Avasimibe

Avasimibe

SCHEMBL15876

CC(C)c1cc(C(C)C)c(CC(=O)NS(=O)(=O)Oc2c(C(C)C)cccc2C(C)C)c(C(C)C)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SOAT2 O75908 1/20 1.00
MYC P01106 1/20 1.00
SOAT1 P35610 1/20 1.00
MAP2K3 P46734 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24233324 0.93 SOAT2 (0.87) SOAT2MYCSOAT1MAP2K3
SCHEMBL7573425 0.90 SOAT2 (0.81) SOAT2MYCSOAT1MAP2K3
SCHEMBL7567657 0.89 SOAT2 (0.79) SOAT2MYCSOAT1MAP2K3
SCHEMBL7612729 0.88 SOAT2 (0.79) SOAT2MYCSOAT1MAP2K3
SCHEMBL7567505 0.88 SOAT2 (0.78) SOAT2MYCSOAT1MAP2K3
SCHEMBL7572791 0.88 SOAT2 (0.78) SOAT2MYCSOAT1MAP2K3
SCHEMBL7570156 0.87 SOAT2 (0.77) SOAT2MYCSOAT1MAP2K3
SCHEMBL7565721 0.87 SOAT2 (0.77) SOAT2MYCSOAT1MAP2K3
SCHEMBL7566055 0.87 SOAT2 (0.77) SOAT2MYCSOAT1MAP2K3
SCHEMBL7574340 0.87 SOAT2 (0.77) SOAT2MYCSOAT1MAP2K3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 10722 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026087680-A1 TREATMENT FOR CARDIOVASCULAR DISEASE SAPREME TECHNOLOGIES B.V. (NL) 2026-04-30 WO claimed
US-20260091010-A1 COMPOSITIONS AND METHODS FOR MANAGING REBOUND OF BODY WEIGHT AND METABOLIC PARAMETERS EFIL BIOSCIENCE INC (KR) 2026-04-02 US claimed
US-20260069593-A1 METHODS FOR TREATING CANCER AMGEN INC (US) 2026-03-12 US claimed
WO-2025226325-A2 IN VITRO SYSTEMS FOR GENERATION OF SKIN EQUIVALENTS AND USES THEREOF AND METHODS FOR DIAGNOSIS AND TREATMENT OF CONNECTIVE TISSUE DISORDERS THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2025-10-30 WO claimed
EP-3787631-B1 MODULATORS OF ORPHAN NUCLEAR RECEPTORS FOR NASH AND OTHER METABOLIC DISORDERS UNIV EMORY (US) 2025-09-10 EP claimed
US-20250255829-A1 Multifunctional Nanoparticles and Uses in Managing Cancer and Cardiovascular Diseases UNIV EMORY (US) 2025-08-14 US claimed
US-12303508-B2 Combinatory treatment strategies of cancer based on RNA polymerase I inhibition THE JOHNS HOPKINS UNIVERSITY (US) 2025-05-20 US claimed
US-12274682-B2 Compositions and methods for controlling food intake of animal PURDUE RESEARCH FOUNDATION (US) 2025-04-15 US claimed
US-12274681-B2 Compositions and methods for reducing skin fat PURDUE RESEARCH FOUNDATION (US) 2025-04-15 US claimed
US-12257217-B2 Compositions and methods for treating hyperphagia in prader-willi syndrome PURDUE RESEARCH FOUNDATION (US) 2025-03-25 US claimed
WO-2001074835-A1 O-GLUCOSYLATED BENZAMIDE SGLT2 INHIBITORS AND METHOD BRISTOL-MYERS SQUIBB COMPANY (US) 2001-10-11 WO claimed
WO-2001068603-A2 CYCLOPROPYL-FUSED PYRROLIDINE-BASED INHIBITORS OF DIPEPTIDYL IV, PROCESSES FOR THEIR PREPARATION, AND THEIR USE BRISTOL-MYERS SQUIBB CO. (US) 2001-09-20 WO claimed
WO-2001060807-A1 ARYLOXYACETIC ACIDS FOR DIABETES AND LIPID DISORDERS MERCK & CO. INC. (US) 2001-08-23 WO claimed
WO-2001056556-A2 DUAL INHIBITORS OF CHOLESTERYL ESTER AND WAX ESTER SYNTHESIS FOR SEBACEOUS GLAND DISORDERS WARNER-LAMBERT COMPANY (US) 2001-08-09 WO claimed
EP-1098662-A2 COADMINISTRATION OF ACAT AND MMP INHIBITORS FOR THE TREATMENT OF ATHEROSCLEROTIC LESIONS WARNER-LAMBERT COMPANY (US) 2001-05-16 EP claimed
WO-2001027107-A2 HETEROCYCLIC SODIUM/PROTON EXCHANGE INHIBITORS AND METHOD BRISTOL-MYERS SQUIBB COMPANY (US) 2001-04-19 WO claimed
WO-2001027128-A1 C-ARYL GLUCOSIDE SGLT2 INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2001-04-19 WO claimed
WO-2001021602-A1 OXA- AND THIAZOLE DERIVATIVES USEFUL AS ANTIDIABETIC AND ANTIOBESITY AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2001-03-29 WO claimed
WO-2000059506-A1 HETEROCYCLIC CONTAINING BIPHENYL aP2 INHIBITORS AND METHOD BRISTOL-MYERS SQUIBB CO. (US) 2000-10-12 WO claimed
WO-2000004892-A2 COADMINISTRATION OF ACAT AND MMP INHIBITORS FOR THE TREATMENT OF ATHEROSCLEROTIC LESIONS WARNER-LAMBERT COMPANY (US) 2000-02-03 WO claimed