SCHEMBL15876355

SCHEMBL15876355

CN(C)Cc1ccc(NC(=O)c2cccc(C(N)=O)c2)cc1

nearest known ligand 0.72

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 10/20 0.72
CYP3A4 P08684 2/20 0.59
PLAU P00749 1/20 0.58
CYP2C19 P33261 1/20 0.54
MEN1 O00255 4/20 0.50
KMT2A Q03164 4/20 0.50
TP53 P04637 2/20 0.50
FFAR1 O14842 1/20 0.50
GLA P06280 1/20 0.50
KDM4E B2RXH2 1/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL307838 0.91 ROCK2 (0.81) ROCK2CYP3A4PLAUCYP2C19
SCHEMBL307678 0.85 ROCK2 (0.67) ROCK2CYP3A4PLAUCYP2C19MEN1
SCHEMBL307307 0.85 ROCK2 (0.86) ROCK2CYP3A4CYP2C19MEN1KMT2A
SCHEMBL7242305 0.85 PLAU (0.62) ROCK2PLAUMEN1KMT2ATP53
SCHEMBL10159840 0.84 ROCK2 (1.00) ROCK2CYP3A4CYP2C19
SCHEMBL10159692 0.84 ROCK2 (1.00) ROCK2CYP3A4PLAUCYP2C19
SCHEMBL10160403 0.84 ROCK2 (0.65) ROCK2CYP3A4PLAUCYP2C19MEN1
SCHEMBL15651634 0.82 ROCK2 (0.56) ROCK2CYP3A4CYP2C19MEN1KMT2A
SCHEMBL8546973 0.81 MEN1 (0.53) ROCK2CYP3A4PLAUMEN1KMT2A
SCHEMBL7234090 0.80 NPC1 (0.65) PLAUMEN1KMT2ATP53FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114869-B1 RHO KINASE INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2014-07-23 EP claimed