SCHEMBL15880484

SCHEMBL15880484

CSc1ncc2c(n1)CCN(C(=O)OC(C)(C)C)C2=O

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCNA2 P20248 9/20 0.52
CDK2 P24941 9/20 0.52
MAPT P10636 2/20 0.37
PIM1 P11309 1/20 0.37
PIM2 Q9P1W9 1/20 0.37
HTR2A P28223 1/20 0.36
BUB1 O43683 1/20 0.34
ELANE P08246 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
PLK1 P53350 1/20 0.33
DDB1 Q16531 1/20 0.32
CRBN Q96SW2 1/20 0.32
CKS1B P61024 1/20 0.32
SKP1 P63208 1/20 0.32
SKP2 Q13309 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30294180 1.00 CCNA2 (0.52) CCNA2CDK2MAPTPIM1PIM2
SCHEMBL29964392 0.83 MAPT (0.38) CCNA2CDK2MAPTPIM1PIM2
SCHEMBL28948723 0.83 CCNA2 (0.41) CCNA2CDK2PIM1PIM2HTR2A
SCHEMBL31584245 0.79 CCNA2 (0.44) CCNA2CDK2MAPTHTR2AMEN1
SCHEMBL31584251 0.76 CCNA2 (0.42) CCNA2CDK2MAPTHTR2AMEN1
SCHEMBL785706 0.75 MAPT (0.63) CCNA2CDK2MAPTDDB1CRBN
SCHEMBL12497878 0.75 CCNA2 (0.51) CCNA2CDK2MAPTHTR2ADDB1
SCHEMBL3400140 0.75 PIM1 (0.40) MAPTPIM1PIM2BUB1MEN1
SCHEMBL30684862 0.75 PIM1 (0.40) MAPTPIM1PIM2BUB1MEN1
SCHEMBL18743044 0.74 GRM5 (0.43) CCNA2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025103367-A1 LIGAND-DRUG CONJUGATE, LINKER FOR CONJUGATION, AND USE THEREOF 海南先声再明医药股份有限公司 2025-05-22 WO disclosed
US-20230123268-A1 AMINO-PYRIMIDINE CYCLO-AMIDES HOFFMANN-LA ROCHE INC. (US) 2023-04-20 US disclosed
US-20230123268-A1 AMINO-PYRIMIDINE CYCLO-AMIDES HOFFMANN-LA ROCHE INC. (US) 2023-04-20 US disclosed
EP-4161928-A2 AMINO-PYRIMIDINE CYCLO-AMIDES F. Hoffmann-La Roche AG (CH) 2023-04-12 EP disclosed
EP-3478685-B1 CHIRAL HETEROCYCLIC COMPOUND WITH HEDGEHOG PATHWAY ANTAGONIST ACTIVITY, METHOD AND USE THEREOF SUZHOU KINTOR PHARMACEUTICALS INC (CN) 2022-01-12 EP disclosed
EP-3478685-B1 CHIRAL HETEROCYCLIC COMPOUND WITH HEDGEHOG PATHWAY ANTAGONIST ACTIVITY, METHOD AND USE THEREOF SUZHOU KINTOR PHARMACEUTICALS INC (CN) 2022-01-12 EP disclosed
WO-2021249904-A2 AMINO-PYRIMIDINE CYCLO-AMIDES F. HOFFMANN-LA ROCHE AG (CH) 2021-12-16 WO disclosed
WO-2021249904-A2 AMINO-PYRIMIDINE CYCLO-AMIDES F. HOFFMANN-LA ROCHE AG (CH) 2021-12-16 WO disclosed
US-10919889-B2 Chiral heterocyclic compound with hedgehog pathway antagonist activity, method and use thereof SUZHOU KINTOR PHARMACEUTICALS, INC. (CN) 2021-02-16 US disclosed
US-10919889-B2 Chiral heterocyclic compound with hedgehog pathway antagonist activity, method and use thereof SUZHOU KINTOR PHARMACEUTICALS, INC. (CN) 2021-02-16 US disclosed
EP-2945623-B1 HEDGEHOG PATHWAY SIGNALING INHIBITORS AND THERAPEUTIC APPLICATIONS THEREOF SUZHOU KINTOR PHARMACEUTICALS INC (CN) 2018-09-05 EP disclosed
US-9695178-B2 6-(2-pyridyl)-7,8-dihydro-5H-pyrido[4,3-D]pyrimidine analogs as hedgehog pathway signaling inhibitors and therapeutic applications thereof SUZHOU KINTOR PHARMACEUTICALS, INC. (CN) 2017-07-04 US disclosed
US-9695178-B2 6-(2-pyridyl)-7,8-dihydro-5H-pyrido[4,3-D]pyrimidine analogs as hedgehog pathway signaling inhibitors and therapeutic applications thereof SUZHOU KINTOR PHARMACEUTICALS, INC. (CN) 2017-07-04 US disclosed
US-9695178-B2 6-(2-pyridyl)-7,8-dihydro-5H-pyrido[4,3-D]pyrimidine analogs as hedgehog pathway signaling inhibitors and therapeutic applications thereof SUZHOU KINTOR PHARMACEUTICALS, INC. (CN) 2017-07-04 US disclosed
US-20160024095-A1 HEDGEHOG PATHWAY SIGNALING INHIBITORS AND THERAPEUTIC APPLICATIONS THEREOF SUZHOU KINTOR PHARMACEUTICALS, INC. (CN) 2016-01-28 US disclosed
US-20160024095-A1 HEDGEHOG PATHWAY SIGNALING INHIBITORS AND THERAPEUTIC APPLICATIONS THEREOF SUZHOU KINTOR PHARMACEUTICALS, INC. (CN) 2016-01-28 US disclosed
US-20160024095-A1 HEDGEHOG PATHWAY SIGNALING INHIBITORS AND THERAPEUTIC APPLICATIONS THEREOF SUZHOU KINTOR PHARMACEUTICALS, INC. (CN) 2016-01-28 US disclosed
EP-2945623-A1 HEDGEHOG PATHWAY SIGNALING INHIBITORS AND THERAPEUTIC APPLICATIONS THEREOF Suzhou yunxuan yiyaokeji youxiangongsi (Su Zhou Yuan Pharm) (CN) 2015-11-25 EP disclosed
WO-2014113191-A1 HEDGEHOG PATHWAY SIGNALING INHIBITORS AND THERAPEUTIC APPLICATIONS THEREOF ZHANG XIAOHU (CN) 2014-07-24 WO disclosed
WO-2014113191-A1 HEDGEHOG PATHWAY SIGNALING INHIBITORS AND THERAPEUTIC APPLICATIONS THEREOF ZHANG XIAOHU (CN) 2014-07-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230123268-A1 AMINO-PYRIMIDINE CYCLO-AMIDES ATXN2, ATXN2L, ATXN10 CCNA2 36/4885CDK2 8/4885MAPT 1860/4885
US-20160024095-A1 HEDGEHOG PATHWAY SIGNALING INHIBITORS AND THERAPEUTIC APPLICATIONS THEREOF SHH, GLI1, SMO CCNA2 3162/4885CDK2 1488/4885MAPT 3091/4885
US-10919889-B2 Chiral heterocyclic compound with hedgehog pathway antagonist activity, method and use thereof SHH, GLI1, SMO CCNA2 1464/4885CDK2 427/4885MAPT 4181/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.