SCHEMBL15880641

SCHEMBL15880641

COc1ccccc1C(=O)N(C)C1COC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.47
SLC6A4 P31645 1/20 0.47
KCNH2 Q12809 1/20 0.47
TRPM8 Q7Z2W7 1/20 0.44
TSHR P16473 2/20 0.43
HPGD P15428 1/20 0.43
PDE2A O00408 1/20 0.43
CTSD P07339 1/20 0.43
GAA P10253 1/20 0.42
MAPK1 P28482 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
DRD2 P14416 1/20 0.41
STAT3 P40763 1/20 0.41
FAAH O00519 1/20 0.41
CNR2 P34972 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30514761 0.86 NPC1 (0.52) SLC6A2SLC6A4KCNH2TRPM8TSHR
SCHEMBL30804744 0.80 TSHR (0.47) SLC6A2SLC6A4KCNH2TSHRHPGD
SCHEMBL10107580 0.80 SLC6A4 (0.64) SLC6A2SLC6A4KCNH2TRPM8TSHR
SCHEMBL10293552 0.79 POLB (0.51) SLC6A2SLC6A4KCNH2TSHRHPGD
Hydrochloric Acid SCHEMBL30956785 0.78 POLB (0.53) SLC6A2SLC6A4KCNH2TSHRHPGD
SCHEMBL2541558 0.76 CTSD (0.55) PDE2ACTSDNPC1RAB9AL3MBTL1
SCHEMBL4661421 0.75 HPGD (0.49) SLC6A2SLC6A4KCNH2TRPM8TSHR
SCHEMBL30804741 0.74 USP30 (0.44) TSHRHPGDNPC1RAB9AL3MBTL1
SCHEMBL24634050 0.74 HTT (0.53) HPGDPDE2ACTSDNPC1RAB9A
SCHEMBL10107578 0.73 KDM4E (0.60) KCNH2TSHRMAPK1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2945636-A2 SUBSTITUTED PYRROLOPYRIMIDINE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH Signal Pharmaceuticals, LLC (US) 2015-11-25 EP disclosed
WO-2014113429-A2 SUBSTITUTED PYRROLOPYRIMIDINE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH SIGNAL PHARMACEUTICALS, LLC (US) 2014-07-24 WO disclosed