SCHEMBL15902240

SCHEMBL15902240

CC(C)(C)[Si](C)(C)OCCOc1ccc2c(C(=O)C(Cl)c3ccccc3)c[nH]c2c1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.52
MEN1 O00255 1/20 0.52
HAT1 O14929 4/20 0.44
EP300 Q09472 4/20 0.44
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 1/20 0.41
MDH2 P40926 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAPT P10636 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15902036 0.87 KMT2A (0.57) KMT2AMEN1HAT1EP300CYP2C9
SCHEMBL15901962 0.82 CYP2C9 (0.57) HAT1EP300CYP2C9CYP2C19MAPT
SCHEMBL15902043 0.79 KMT2A (0.54) KMT2AMEN1HAT1EP300CYP2C9
SCHEMBL15902301 0.74 KMT2A (0.49) KMT2AMEN1HAT1EP300CYP2C9
SCHEMBL15902158 0.74 MEN1 (0.49) KMT2AMEN1HAT1EP300ALDH1A1
SCHEMBL15901825 0.73 KMT2A (0.71) KMT2AMEN1HAT1EP300ALDH1A1
SCHEMBL15902547 0.72 KMT2A (0.72) KMT2AMEN1HAT1EP300ALDH1A1
SCHEMBL15902147 0.72 KMT2A (0.67) KMT2AMEN1HAT1EP300ALDH1A1
SCHEMBL15902047 0.71 KMT2A (0.71) KMT2AMEN1HAT1EP300ALDH1A1
SCHEMBL14496307 0.70 KMT2A (1.00) KMT2AMEN1HAT1EP300ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12012411-B2 Viral replication inhibitors KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2024-06-18 US disclosed
US-20220106321-A1 VIRAL REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2022-04-07 US disclosed
US-11279704-B2 Viral replication inhibitors KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2022-03-22 US disclosed
CN-108440370-B Inhibitors of viral replication 鲁汶天主教大学 2021-07-30 CN disclosed
EP-3617192-A1 VIRAL REPLICATION INHIBITORS Katholieke Universiteit Leuven K.U. Leuven R&D (BE) 2020-03-04 EP disclosed
US-10550123-B2 Viral replication inhibitors KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2020-02-04 US disclosed
US-20190337954-A1 VIRAL REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2019-11-07 US disclosed
EP-2760831-B1 VIRAL REPLICATION INHIBITORS UNIV LEUVEN KATH (BE) 2019-08-07 EP disclosed
US-20140213586-A1 VIRAL REPLICATION INHIBITORS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2014-07-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140213586-A1 VIRAL REPLICATION INHIBITORS EIF2AK2, MAVS, ZC3HAV1 KMT2A 2425/4885MEN1 3390/4885HAT1 3301/4885
US-11279704-B2 Viral replication inhibitors EIF2AK2, MAVS, ZC3HAV1 KMT2A 2425/4885MEN1 3390/4885HAT1 3301/4885
US-20190337954-A1 VIRAL REPLICATION INHIBITORS EIF2AK2, MAVS, ZC3HAV1 KMT2A 2425/4885MEN1 3390/4885HAT1 3301/4885
US-10550123-B2 Viral replication inhibitors EIF2AK2, MAVS, ZC3HAV1 KMT2A 2425/4885MEN1 3390/4885HAT1 3301/4885
US-20220106321-A1 VIRAL REPLICATION INHIBITORS EIF2AK2, MAVS, ZC3HAV1 KMT2A 2425/4885MEN1 3390/4885HAT1 3301/4885
US-12012411-B2 Viral replication inhibitors EIF2AK2, MAVS, ZC3HAV1 KMT2A 2425/4885MEN1 3390/4885HAT1 3301/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.