SCHEMBL15902805

SCHEMBL15902805

COc1ccc(CN[N+]23C=CN=CC2=C(C2CCC(CO)N(C(=O)OCc4ccccc4)C2)N=C3c2ccc(C(=O)Nc3cc(C(F)(F)F)ccn3)cc2)c(OC)c1

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BTK Q06187 18/20 0.36
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15903372 0.91 BTK (0.37) BTK
SCHEMBL15877657 0.84 BTK (0.37) BTK
SCHEMBL15877499 0.82 BTK (0.47) BTK
SCHEMBL15878595 0.82 BTK (0.47) BTK
SCHEMBL15878807 0.81 BTK (0.33) BTK
SCHEMBL15904443 0.80 BTK (0.45) BTK
SCHEMBL15877670 0.79 BTK (0.34) BTK
SCHEMBL15913882 0.78 ALDH1A1 (0.40) ALDH1A1TP53
SCHEMBL15878328 0.77 BTK (0.50) BTK
SCHEMBL14637752 0.76 ALDH1A1 (0.39) ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014113932-A1 BTK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2014-07-31 WO disclosed