SCHEMBL15903294

SCHEMBL15903294

CCOCCON(C(=O)c1ccccc1)c1cc(C(F)(F)F)ccn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.42
ALDH1A1 P00352 3/20 0.39
GAA P10253 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
POLQ O75417 2/20 0.39
OPRM1 P35372 1/20 0.38
OPRL1 P41146 1/20 0.38
HTT P42858 1/20 0.38
PTGDR2 Q9Y5Y4 2/20 0.36
VCP P55072 1/20 0.35
GLA P06280 1/20 0.35
HPGD P15428 1/20 0.35
CNR2 P34972 2/20 0.35
TRPA1 O75762 1/20 0.35
CYP1A2 P05177 1/20 0.35
TBXA2R P21731 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
TAAR1 Q96RJ0 1/20 0.35
LIPG Q9Y5X9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17892578 0.90 MAPK14 (0.45) MAPK14ALDH1A1GAAL3MBTL1POLQ
SCHEMBL15903436 0.89 HTT (0.48) MAPK14ALDH1A1GAAL3MBTL1POLQ
SCHEMBL15903063 0.87 MAPK14 (0.40) MAPK14GAAPOLQOPRM1OPRL1
SCHEMBL15903204 0.84 MAPK14 (0.41) MAPK14ALDH1A1GAAL3MBTL1POLQ
SCHEMBL18825315 0.82 HTT (0.40) MAPK14GAAPOLQOPRM1OPRL1
SCHEMBL17894004 0.81 MAPK14 (0.41) MAPK14ALDH1A1GAAL3MBTL1POLQ
SCHEMBL15903268 0.78 MAPK14 (0.39) MAPK14POLQOPRM1OPRL1HTT
SCHEMBL15903361 0.74 ALDH1A1 (0.41) MAPK14ALDH1A1GAAOPRM1OPRL1
SCHEMBL15903091 0.73 GLA (0.41) MAPK14GAAPOLQOPRM1OPRL1
SCHEMBL17894096 0.73 ALDH1A1 (0.36) MAPK14ALDH1A1GAAL3MBTL1POLQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2948458-A1 BTK INHIBITORS Merck Sharp & Dohme Corp. (US) 2015-12-02 EP claimed
WO-2014114185-A1 BTK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2014-07-31 WO claimed
EP-2948458-A1 BTK INHIBITORS Merck Sharp & Dohme Corp. (US) 2015-12-02 EP disclosed
WO-2014114185-A1 BTK INHIBITORS MERCK SHARP & DOHME CORP. (US) 2014-07-31 WO disclosed