Ibezapolstat

Ibezapolstat

SCHEMBL15908884

O=c1[nH]c(NCc2ccc(Cl)c(Cl)c2)nc2ncn(CCN3CCOCC3)c12

nearest known ligand 0.00

Full drug profile on Sugi Atlas →

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ibezapolstat SCHEMBL29357391 1.00
Ibezapolstat SCHEMBL15908913 0.99
SCHEMBL12173570 0.95
SCHEMBL1443265 0.95
Hydrochloric Acid SCHEMBL15909144 0.95
SCHEMBL1443301 0.95
Hydrochloric Acid SCHEMBL1443775 0.95
Hydrochloric Acid SCHEMBL1443761 0.94
SCHEMBL1443553 0.93
SCHEMBL1443493 0.89

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8796292-B2 Selective antibacterials for clostridium difficile infections GLSYNTHESIS INC. (US) 2014-08-05 US claimed
US-20240316058-A1 Use of Ibezapolstat to Promote Microbiome Health Acurx Pharmaceuticals, Inc. 2024-09-26 US disclosed
US-12036225-B2 Use of ibezapolstat to promote microbiome health Acurx Pharmaceuticals, Inc. (US) 2024-07-16 US disclosed
CN-117813085-A Use of Bei Zabo erstat for promoting microbiome health 阿科利斯制药股份有限公司 2024-04-02 CN disclosed
EP-4340827-A2 USE OF IBEZAPOLSTAT TO PROMOTE MICROBIOME HEALTH Acurx Pharmaceuticals, Inc. (US) 2024-03-27 EP disclosed
US-20220409625-A1 Use of Ibezapolstat to Promote Microbiome Health Acurx Pharmaceuticals, Inc. 2022-12-29 US disclosed
WO-2022266318-A2 USE OF IBEZAPOLSTAT TO PROMOTE MICROBIOME HEALTH ACURX PHARMACEUTICALS LLC (US) 2022-12-22 WO disclosed
US-20220024925-A1 Deuterium-Substituted 7-Substituted-2-(Benzylamino)-6-Ozopurine Compounds and Uses Thereof ACURX PHARMACEUTICALS, LLC 2022-01-27 US disclosed