SCHEMBL15911397

SCHEMBL15911397

Cc1cc(C)n(C(=O)CN2CCN(c3ccccc3-c3cnc(N4CCC(S(C)(=O)=O)CC4)nc3)CC2C)n1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 5/20 0.41
KCNH2 Q12809 1/20 0.41
GAA P10253 1/20 0.36
HTR1A P08908 2/20 0.35
DRD2 P14416 2/20 0.35
HTR7 P34969 2/20 0.35
HTR6 P50406 2/20 0.35
WDR5 P61964 5/20 0.35
ALDH1A1 P00352 3/20 0.34
TSHR P16473 1/20 0.34
SLC6A9 P48067 1/20 0.34
MAPT P10636 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
TP53 P04637 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15911221 0.91 CXCR3 (0.37) CXCR3WDR5
SCHEMBL15911228 0.89 CXCR3 (0.40) CXCR3KCNH2WDR5ALDH1A1
SCHEMBL163847 0.85 CXCR3 (0.50) CXCR3KCNH2
SCHEMBL3730941 0.80 CXCR3 (0.66) CXCR3KCNH2GAAALDH1A1TSHR
SCHEMBL15911460 0.79 CXCR3 (0.41) CXCR3KCNH2WDR5
SCHEMBL166781 0.76 CXCR3 (0.52) CXCR3KCNH2
SCHEMBL15911340 0.76 CXCR3 (0.51) CXCR3KCNH2GAADRD2ALDH1A1
SCHEMBL165663 0.75 CXCR3 (0.53) CXCR3KCNH2
SCHEMBL111968 0.74 CXCR3 (0.37) CXCR3KCNH2ALDH1A1
SCHEMBL165135 0.74 CXCR3 (0.55) CXCR3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424840-B1 CXCR3 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2014-08-06 EP disclosed