SCHEMBL1591176

SCHEMBL1591176

NC(=O)[C@H](O)[C@H](O)[C@H](O)CO

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.52
LMNA P02545 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
USP2 O75604 1/20 0.48
SLCO1B1 Q9Y6L6 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
PGD P52209 1/20 0.39
KDM4E B2RXH2 2/20 0.36
TGFBR1 P36897 1/20 0.32
OR51E2 Q9H255 1/20 0.32
CYP2C9 P11712 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL122819 1.00 PDE4A (0.52) PDE4ALMNAL3MBTL1USP2SLCO1B1
SCHEMBL4728437 1.00 PDE4A (0.52) PDE4ALMNAL3MBTL1USP2SLCO1B1
SCHEMBL4638447 1.00 PDE4A (0.52) PDE4ALMNAL3MBTL1USP2SLCO1B1
SCHEMBL2126263 1.00 PDE4A (0.52) PDE4ALMNAL3MBTL1USP2SLCO1B1
SCHEMBL7151302 1.00 PDE4A (0.52) PDE4ALMNAL3MBTL1USP2SLCO1B1
SCHEMBL6665411 1.00 PDE4A (0.52) PDE4ALMNAL3MBTL1USP2SLCO1B1
SCHEMBL1569332 0.92 PDE4A (0.62) PDE4ALMNAL3MBTL1USP2SLCO1B1
SCHEMBL5268306 0.92 PDE4A (0.62) PDE4ALMNAL3MBTL1USP2SLCO1B1
SCHEMBL2912046 0.92 PDE4A (0.62) PDE4ALMNAL3MBTL1USP2SLCO1B1
SCHEMBL20576207 0.92 PDE4A (0.62) PDE4ALMNAL3MBTL1USP2SLCO1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 150 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025111452-A2 CHEMICAL MODIFICATIONS IN PEgRNA and ngRNAs PRIME MEDICINE, INC. (US) 2025-05-30 WO claimed
WO-2025111430-A1 CHEMICAL MODIFICATIONS IN mRNA POLY(A) TAIL PRIME MEDICINE, INC. (US) 2025-05-30 WO claimed
WO-2025038960-A1 OLIGONUCLEOTIDES CONTAINING A LIGAND AT AN INTERNAL POSITION ADARX PHARMACEUTICALS, INC. (US) 2025-02-20 WO claimed
CN-119095964-A Multi-tail and multi-cap mRNA and uses thereof 博德研究所 2024-12-06 CN claimed
EP-4466074-A1 POLY-TAILED AND POLY-CAPPED MRNA AND USES THEREOF The Broad Institute Inc. (US) 2024-11-27 EP claimed
EP-4337331-A1 MODIFIED MRNA, MODIFIED NON-CODING RNA, AND USES THEREOF The Broad Institute Inc. (US) 2024-03-20 EP claimed
WO-2023141474-A9 POLY-TAILED AND POLY-CAPPED MRNA AND USES THEREOF THE BROAD INSTITUTE, INC. (US) 2023-10-26 WO claimed
WO-2023141474-A1 POLY-TAILED AND POLY-CAPPED MRNA AND USES THEREOF THE BROAD INSTITUTE, INC. (US) 2023-07-27 WO claimed
WO-2022241045-A1 MODIFIED MRNA, MODIFIED NON-CODING RNA, AND USES THEREOF THE BROAD INSTITUTE, INC. (US) 2022-11-17 WO claimed
CN-114729355-A PPM1A inhibitors and methods of using the same 奎里斯公司 2022-07-08 CN claimed
US-8541567-B2 Transition state structure of 5′-methylthioadenosine/s-adenosylhomocysteine nucleosidases ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2013-09-24 US claimed
US-20110086812-A1 Transition state sturcture of 5'-methylthioadenosine/s-adenosylhomocysteine nucleosidases ALBERT EINSTEIN COLLEGE OF MEDICINE 2011-04-14 US claimed
US-20100062995-A1 Transition state structure of human 5'methylthioadenosine phosphorylase NATIONAL INSTITUTES OF HEALTH 2010-03-11 US claimed
EP-2066671-A1 TRANSITION STATE STRUCTURE OF HUMAN 5'-METHYLTHIOADENOSINE PHOSPHORYLASE ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2009-06-10 EP claimed
EP-1924684-A4 TRANSITION STATE STRUCTURE OF 5'-METHYLTHIOADENOSINE/S-ADENOSYLHOMOCYSTEINE NUCLEOSIDASES EINSTEIN COLL MED (US) 2009-02-11 EP claimed
EP-1924684-A2 TRANSITION STATE STRUCTURE OF 5'-METHYLTHIOADENOSINE/S-ADENOSYLHOMOCYSTEINE NUCLEOSIDASES ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY, a division of YESHIVA UNIVERSITY (US) 2008-05-28 EP claimed
WO-2008039324-A1 TRANSITION STATE STRUCTURE OF HUMAN 5'-METHYLTHIOADENOSINE PHOSPHORYLASE ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2008-04-03 WO claimed
WO-2007016291-A2 TRANSITION STATE STRUCTURE OF 5'-METHYLTHIOADENOSINE/S-ADENOSYLHOMOCYSTEINE NUCLEOSIDASES ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2007-02-08 WO claimed
EP-0946744-A1 NOVEL POLYMERIC COMPLEXES FOR THE TRANSFECTION OF NUCLEIC ACIDS, WITH RESIDUES CAUSING THE DESTABILISATION OF CELL MEMBRANES I.D.M. IMMUNO-DESIGNED MOLECULES (FR) 1999-10-06 EP claimed
WO-1998022610-A1 NOVEL POLYMERIC COMPLEXES FOR THE TRANSFECTION OF NUCLEIC ACIDS, WITH RESIDUES CAUSING THE DESTABILISATION OF CELL MEMBRANES I.D.M. IMMUNO-DESIGNED MOLECULES (FR) 1998-05-28 WO claimed