SCHEMBL15918593

SCHEMBL15918593

NOCCCOc1ccc(Br)nc1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.40
CHRNA4 P43681 2/20 0.40
TMPRSS2 O15393 1/20 0.35
FURIN P09958 1/20 0.34
PRSS1 P07477 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16451529 0.81 TAAR1 (0.47) CHRNB2CHRNA4
SCHEMBL20577124 0.81 CHRNB2 (0.42) CHRNB2CHRNA4
SCHEMBL30692795 0.81 CHRNB2 (0.42) CHRNB2CHRNA4
SCHEMBL20577017 0.81 CHRNB2 (0.42) CHRNB2CHRNA4
SCHEMBL1109106 0.81 CYP2D6 (0.47) CHRNB2CHRNA4
SCHEMBL30692819 0.81 CHRNB2 (0.42) CHRNB2CHRNA4
SCHEMBL15901278 0.79 CHRNB2 (0.41) CHRNB2CHRNA4
SCHEMBL15082431 0.79 MAPT (0.44) CHRNB2CHRNA4
Hydrochloric Acid SCHEMBL16332831 0.79 TAAR1 (0.45) CHRNB2CHRNA4
SCHEMBL17658773 0.79 CHRNB2 (0.43) CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014114578-A1 PYRROLIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-07-31 WO disclosed