SCHEMBL15922228

SCHEMBL15922228

O=C(NC(Nc1ccc2ccccc2c1)C(Cl)(Cl)Cl)c1ccco1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 14/20 0.55
MAPT P10636 9/20 0.55
KMT2A Q03164 8/20 0.55
MEN1 O00255 7/20 0.55
LMNA P02545 5/20 0.55
NPSR1 Q6W5P4 5/20 0.54
ALOX12 P18054 2/20 0.54
PKM P14618 1/20 0.54
HTT P42858 2/20 0.51
GAA P10253 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
L3MBTL1 Q9Y468 1/20 0.50
KDM4E B2RXH2 2/20 0.49
HPGD P15428 2/20 0.49
POLB P06746 1/20 0.49
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1923366 0.83 ALDH1A1 (0.72) ALDH1A1MAPTKMT2AMEN1LMNA
SCHEMBL1923000 0.81 ALDH1A1 (0.73) ALDH1A1MAPTKMT2AMEN1LMNA
SCHEMBL1923376 0.81 ALDH1A1 (0.58) ALDH1A1MAPTKMT2AMEN1LMNA
SCHEMBL12156722 0.81 NPC1 (0.58) ALDH1A1MAPTKMT2AMEN1LMNA
SCHEMBL1923694 0.81 ALDH1A1 (0.61) ALDH1A1MAPTKMT2AMEN1LMNA
SCHEMBL1923385 0.81 ALDH1A1 (0.56) ALDH1A1MAPTKMT2AMEN1LMNA
SCHEMBL1923002 0.81 ALDH1A1 (0.56) ALDH1A1MAPTKMT2AMEN1LMNA
SCHEMBL6669056 0.76 SMN1; SMN2 (0.75) ALDH1A1MAPTKMT2AMEN1LMNA
SCHEMBL1922861 0.76 KMT2A (0.60) ALDH1A1MAPTKMT2AMEN1LMNA
SCHEMBL1923358 0.74 ALDH1A1 (0.61) ALDH1A1MAPTKMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014120790-A1 SMALL MOLECULES TO BLOCK SIGNALING PATHWAY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2014-08-07 WO claimed
WO-2014120790-A1 SMALL MOLECULES TO BLOCK SIGNALING PATHWAY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2014-08-07 WO disclosed
WO-2014120790-A1 SMALL MOLECULES TO BLOCK SIGNALING PATHWAY THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2014-08-07 WO disclosed