SCHEMBL15925501

SCHEMBL15925501

CNc1ccc(-c2ccccc2N2CCN(C(=O)Cn3nc(C)cc3C)CC2)cc1

nearest known ligand 0.83

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 3/20 0.83
KCNH2 Q12809 1/20 0.83
ALDH1A1 P00352 3/20 0.47
LMNA P02545 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.42
KMT2A Q03164 1/20 0.42
TSHR P16473 1/20 0.41
MGLL Q99685 1/20 0.41
DPP4 P27487 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3732781 0.91 CXCR3 (0.78) CXCR3KCNH2ALDH1A1LMNASMN1; SMN2
SCHEMBL3732650 0.91 CXCR3 (0.96) CXCR3KCNH2ALDH1A1LMNAKMT2A
SCHEMBL3730735 0.91 CXCR3 (0.88) CXCR3KCNH2ALDH1A1LMNASMN1; SMN2
SCHEMBL3735739 0.91 CXCR3 (0.88) CXCR3KCNH2ALDH1A1LMNAKMT2A
SCHEMBL112559 0.91 CXCR3 (1.00) CXCR3KCNH2ALDH1A1LMNAKMT2A
SCHEMBL114424 0.90 CXCR3 (0.75) CXCR3KCNH2ALDH1A1LMNASMN1; SMN2
SCHEMBL3809576 0.89 CXCR3 (0.78) CXCR3KCNH2ALDH1A1LMNASMN1; SMN2
SCHEMBL3740353 0.89 CXCR3 (0.85) CXCR3KCNH2ALDH1A1LMNAKMT2A
SCHEMBL3726591 0.89 CXCR3 (0.84) CXCR3KCNH2ALDH1A1LMNASMN1; SMN2
SCHEMBL3742966 0.89 CXCR3 (0.84) CXCR3KCNH2ALDH1A1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424840-B1 CXCR3 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2014-08-06 EP disclosed