SCHEMBL15925529

SCHEMBL15925529

CCOc1ncc(-c2cc(F)ccc2N2CCN(C(=O)Cn3ccc4ccncc43)CC2)cn1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 3/20 0.45
KCNH2 Q12809 1/20 0.45
GRIN2B Q13224 15/20 0.44
GRM5 P41594 2/20 0.40
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
GRIN1 Q05586 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL164717 0.93 GRIN2B (0.45) CXCR3GRIN2BGRM5CYP2C9CYP2C19
SCHEMBL3724584 0.87 GRIN2B (0.48) GRIN2BGRM5
SCHEMBL3735698 0.85 GRIN2B (0.49) GRIN2B
SCHEMBL167110 0.84 GRIN2B (0.45) CXCR3KCNH2GRIN2BGRM5
SCHEMBL160222 0.82 GRIN2B (0.40) CXCR3GRIN2BGRM5
SCHEMBL3735612 0.81 GRIN2B (0.42) CXCR3KCNH2GRIN2B
SCHEMBL3735661 0.78 CXCR3 (0.46) CXCR3KCNH2GRIN2BGRM5
SCHEMBL114594 0.75 CXCR3 (0.44) CXCR3KCNH2GRIN2B
SCHEMBL13076636 0.74 SCN10A (0.40) CXCR3GRIN2BGRM5
SCHEMBL3735551 0.72 GRM5 (0.46) CXCR3GRIN2BGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424840-B1 CXCR3 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2014-08-06 EP disclosed