SCHEMBL15925546

SCHEMBL15925546

CC1CN(c2ccccc2-c2cnc([SH](C)(C)=O)nc2)CCN1C(=O)Cn1c(=O)[nH]c2ccccc21

nearest known ligand 0.45

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CXCR3 P49682 18/20 0.45
KCNH2 Q12809 2/20 0.45
LIMK2 P53671 1/20 0.37
HTR7 P34969 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL164924 0.87 CXCR3 (0.47) CXCR3KCNH2LIMK2HTR7
SCHEMBL165175 0.86 CXCR3 (0.62) CXCR3KCNH2LIMK2
SCHEMBL169464 0.85 CXCR3 (0.52) CXCR3KCNH2LIMK2
SCHEMBL15925539 0.80 CXCR3 (0.44) CXCR3KCNH2LIMK2
SCHEMBL167594 0.79 CXCR3 (0.46) CXCR3KCNH2
SCHEMBL113350 0.77 CXCR3 (0.51) CXCR3KCNH2
SCHEMBL15925565 0.77 CXCR3 (0.44) CXCR3KCNH2
SCHEMBL165523 0.77 CXCR3 (0.44) CXCR3KCNH2
SCHEMBL115409 0.76 CXCR3 (0.57) CXCR3KCNH2
SCHEMBL113349 0.75 CXCR3 (0.50) CXCR3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424840-B1 CXCR3 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2014-08-06 EP disclosed