SCHEMBL15925697

SCHEMBL15925697

COC(c1ccc(Cl)cc1)c1cc(-c2ccncc2)sc1-c1ncc[nH]1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.33
GCGR P47871 6/20 0.32
MAPK14 Q16539 4/20 0.32
ROCK1 Q13464 5/20 0.32
CDC7 O00311 4/20 0.32
DBF4 Q9UBU7 4/20 0.32
AKT1 P31749 3/20 0.32
CCNE1 P24864 3/20 0.32
CDK2 P24941 3/20 0.32
SMPD3 Q9NY59 1/20 0.30
FFAR2 O15552 1/20 0.30
LMNA P02545 1/20 0.30
CHRM2 P08172 1/20 0.30
ADRA2B P18089 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
HRH1 P35367 1/20 0.30
SLC6A3 Q01959 1/20 0.30
KCNH2 Q12809 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627649 0.84 ROCK1 (0.32) CYP19A1GCGRMAPK14ROCK1CDC7
SCHEMBL15925726 0.84 CYP19A1 (0.35) CYP19A1GCGRMAPK14ROCK1CDC7
SCHEMBL15925715 0.84 CYP19A1 (0.35) CYP19A1GCGRMAPK14ROCK1CDC7
SCHEMBL15925709 0.84 CYP19A1 (0.35) CYP19A1GCGRMAPK14ROCK1CDC7
SCHEMBL15925751 0.83 CDC7 (0.40) CDC7DBF4FFAR2
SCHEMBL15925691 0.83 CYP19A1 (0.33) CYP19A1GCGRMAPK14ROCK1CDC7
SCHEMBL15925700 0.83 CYP19A1 (0.33) CYP19A1GCGRMAPK14ROCK1CDC7
SCHEMBL15925722 0.83 CYP19A1 (0.33) CYP19A1GCGRMAPK14ROCK1CDC7
SCHEMBL15925718 0.82 AKT1 (0.51) CYP19A1GCGRROCK1CDC7DBF4
SCHEMBL15925714 0.79 SMN1; SMN2 (0.38) CYP19A1ROCK1CDC7DBF4AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8796271-B2 Heteroaryls and uses thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2014-08-05 US disclosed