SCHEMBL15925751

SCHEMBL15925751

COC(c1ccc(Cl)cc1)c1cc(-c2ccnc(NC(C)=O)c2)sc1-c1ncc[nH]1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 1/20 0.40
DBF4 Q9UBU7 1/20 0.40
PIK3C3 Q8NEB9 12/20 0.39
AAK1 Q2M2I8 4/20 0.37
CYP3A4 P08684 2/20 0.37
TGFBR1 P36897 1/20 0.36
TGFBR2 P37173 1/20 0.36
FFAR2 O15552 1/20 0.35
FPR2 P25090 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15925699 0.90 CDC7 (0.43) CDC7DBF4PIK3C3AAK1CYP3A4
SCHEMBL10288582 0.89 CDC7 (0.39) CDC7DBF4PIK3C3AAK1CYP3A4
SCHEMBL15925740 0.89 CDC7 (0.40) CDC7DBF4PIK3C3AAK1CYP3A4
SCHEMBL15925761 0.85 CDC7 (0.41) CDC7DBF4PIK3C3TGFBR1TGFBR2
SCHEMBL15925767 0.84 CDC7 (0.39) CDC7DBF4PIK3C3AAK1CYP3A4
SCHEMBL15925697 0.83 CYP19A1 (0.33) CDC7DBF4FFAR2
SCHEMBL15925763 0.82 CDC7 (0.37) CDC7DBF4PIK3C3AAK1CYP3A4
SCHEMBL15925755 0.80 CDC7 (0.37) CDC7DBF4PIK3C3AAK1CYP3A4
SCHEMBL15925774 0.80 CDC7 (0.37) CDC7DBF4PIK3C3AAK1CYP3A4
SCHEMBL954033 0.79 CDC7 (0.46) CDC7DBF4PIK3C3AAK1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8796271-B2 Heteroaryls and uses thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2014-08-05 US disclosed