SCHEMBL15933429

SCHEMBL15933429

Brc1cccc(-c2cn3c(n2)CNCC3)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.57
CD274 Q9NZQ7 1/20 0.57
TLR9 Q9NR96 1/20 0.46
TLR8 Q9NR97 1/20 0.46
TLR7 Q9NYK1 1/20 0.46
WDR5 P61964 6/20 0.42
ALDH1A1 P00352 4/20 0.41
IDO1 P14902 1/20 0.39
METAP2 P50579 1/20 0.39
RAB9A P51151 2/20 0.39
LMNA P02545 2/20 0.39
HTT P42858 2/20 0.39
KDM4E B2RXH2 1/20 0.39
NPC1 O15118 1/20 0.39
HPGD P15428 3/20 0.38
MAPT P10636 1/20 0.38
HK1 P19367 1/20 0.38
HKDC1 Q2TB90 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15933436 0.84 PDCD1 (0.64) PDCD1CD274TLR9TLR8TLR7
SCHEMBL505942 0.84 PDCD1 (0.57) PDCD1CD274TLR9TLR8TLR7
SCHEMBL15933527 0.84 PDCD1 (0.57) PDCD1CD274TLR9TLR8TLR7
SCHEMBL15933432 0.84 PDCD1 (0.57) PDCD1CD274TLR9TLR8TLR7
SCHEMBL15933525 0.83 PDCD1 (0.52) PDCD1CD274TLR9TLR8TLR7
SCHEMBL108698 0.83 PDCD1 (0.69) PDCD1CD274TLR9TLR8TLR7
SCHEMBL15933694 0.82 PDCD1 (0.55) PDCD1CD274TLR9TLR8TLR7
SCHEMBL15933435 0.81 PDCD1 (0.54) PDCD1CD274TLR9TLR8TLR7
SCHEMBL15933430 0.81 PDCD1 (0.54) PDCD1CD274TLR9TLR8TLR7
SCHEMBL15933431 0.81 WDR5 (0.67) PDCD1CD274TLR9TLR8TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014117318-A1 NOVEL TRIAZOLE ANTIFUNGAL COMPOUNDS, AND PHARMACEUTICAL COMPOSITION, PREPARATION METHOD, AND APPLICATION THEREOF 中国科学院上海药物研究所 (CN) 2014-08-07 WO disclosed