SCHEMBL15935910

SCHEMBL15935910

Cc1ccc2c(c1)CC1(C2)OC(=O)Nc2ncncc21

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 14/20 0.36
ADRA2A P08913 1/20 0.32
KDM4E B2RXH2 2/20 0.30
ALDH1A1 P00352 2/20 0.30
F2 P00734 2/20 0.30
GAA P10253 2/20 0.30
ALOX12 P18054 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13062460 0.85 PARP1 (0.32)
SCHEMBL13015185 0.85 DGAT1 (0.30) AVPR1A
SCHEMBL13747461 0.81 KCNH2 (0.43) AVPR1AALDH1A1GAASMN1; SMN2
SCHEMBL15935915 0.79 AVPR1A (0.38) AVPR1AADRA2AKDM4EALDH1A1F2
SCHEMBL15935911 0.79 CALCRL (0.39) ADRA2AALDH1A1GAASMN1; SMN2
SCHEMBL30032839 0.77 KCNH2 (0.32)
SCHEMBL30033980 0.74
SCHEMBL30032838 0.74 KCNH2 (0.31)
SCHEMBL15935917 0.74 KCNH2 (0.37) SMN1; SMN2
SCHEMBL13747954 0.72 CCNC (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8796260-B2 Imidazobenzazepine CGRP receptor antagonists MERCK SHARP & DOHME CORP. (US) 2014-08-05 US disclosed