SCHEMBL15935945

SCHEMBL15935945

CN1CCC2(CC1)CC(=O)Nc1nccnc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.38
CHRM2 P08172 1/20 0.36
CHRM3 P20309 1/20 0.36
NEK2 P51955 1/20 0.35
HTR2B P41595 3/20 0.35
OPRM1 P35372 1/20 0.35
HTR2A P28223 2/20 0.34
HTR2C P28335 2/20 0.34
SIGMAR1 Q99720 2/20 0.34
CRBN Q96SW2 4/20 0.33
MAPKAPK2 P49137 1/20 0.33
OTUD7B Q6GQQ9 2/20 0.32
DDB1 Q16531 1/20 0.32
BRD4 O60885 1/20 0.32
ATAD2 Q6PL18 1/20 0.32
DRD2 P14416 1/20 0.30
NFKB1 P19838 1/20 0.30
DRD4 P21917 1/20 0.30
BLM P54132 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13748218 0.80 CRBN (0.32) KCNH2NEK2CRBNMAPKAPK2
SCHEMBL1700114 0.78 KCNH2 (0.54) KCNH2CHRM2CHRM3HTR2BHTR2A
SCHEMBL15935916 0.76 FGFR1 (0.38) NEK2HTR2BOPRM1OTUD7BBRD4
SCHEMBL15935940 0.72 KCNH2 (0.38) KCNH2CHRM2CHRM3NEK2HTR2B
SCHEMBL15935948 0.72 CHRM2 (0.36) KCNH2CHRM2CHRM3NEK2HTR2B
SCHEMBL15935918 0.72 KCNH2 (0.39) KCNH2SIGMAR1DRD2
SCHEMBL800500 0.71 CRBN (0.46) CHRM2CHRM3NEK2HTR2BHTR2A
SCHEMBL26141991 0.65 CRBN (0.51) CHRM2CHRM3NEK2CRBNDDB1
SCHEMBL13314948 0.65 PLD1 (0.49) HTR2BHTR2AHTR2CSIGMAR1CRBN
SCHEMBL13342752 0.64 KCNH2 (0.52) KCNH2CHRM2OPRM1CRBNOTUD7B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8796260-B2 Imidazobenzazepine CGRP receptor antagonists MERCK SHARP & DOHME CORP. (US) 2014-08-05 US disclosed