SCHEMBL15935918

SCHEMBL15935918

CN1CCC2(CC1)OC(=O)Nc1nccnc12

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.39
SIGMAR1 Q99720 3/20 0.36
DRD2 P14416 2/20 0.36
PLD2 O14939 1/20 0.35
PLD1 Q13393 1/20 0.35
AVPR1A P37288 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1700113 0.79 KCNH2 (0.55) KCNH2SIGMAR1DRD2AVPR1A
SCHEMBL15935916 0.75 FGFR1 (0.38)
SCHEMBL23508657 0.74 SIGMAR1 (0.35) SIGMAR1DRD2AVPR1A
SCHEMBL15935917 0.73 KCNH2 (0.37) KCNH2SIGMAR1DRD2PLD2PLD1
SCHEMBL15935919 0.73 SIGMAR1 (0.39) KCNH2SIGMAR1DRD2PLD2PLD1
SCHEMBL15935915 0.72 AVPR1A (0.38) KCNH2AVPR1A
SCHEMBL15935945 0.72 KCNH2 (0.38) KCNH2SIGMAR1DRD2
SCHEMBL12175572 0.71 AVPR1A (0.45) SIGMAR1DRD2AVPR1A
SCHEMBL16274418 0.67 SIGMAR1 (0.47) SIGMAR1DRD2
SCHEMBL1700111 0.66 TP53 (0.56) SIGMAR1DRD2PLD2PLD1AVPR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8796260-B2 Imidazobenzazepine CGRP receptor antagonists MERCK SHARP & DOHME CORP. (US) 2014-08-05 US disclosed