SCHEMBL15936941

SCHEMBL15936941

Cc1c(C(=O)N2CCCC(=O)N([C@H](C(N)=O)[C@@H](C)O)C2)nnn1Cc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.38
KLKB1 P03952 1/20 0.37
CYP19A1 P11511 4/20 0.37
CYP1A2 P05177 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
LMNA P02545 3/20 0.35
POLB P06746 1/20 0.35
EEF2K O00418 1/20 0.35
DRD2 P14416 4/20 0.35
DRD4 P21917 4/20 0.35
DRD3 P35462 4/20 0.35
HTR2A P28223 3/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA3 P07451 1/20 0.35
CA4 P22748 1/20 0.35
CA6 P23280 1/20 0.35
CA5A P35218 1/20 0.35
CA7 P43166 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19229626 0.78 GRIN2B (0.49) HPGDKLKB1CYP19A1CYP1A2SMN1; SMN2
SCHEMBL17712366 0.78 GRIN2B (0.49) HPGDKLKB1CYP19A1CYP1A2SMN1; SMN2
SCHEMBL20485072 0.78 GRIN2B (0.49) HPGDKLKB1CYP19A1CYP1A2SMN1; SMN2
SCHEMBL21467087 0.75 CYP19A1 (0.39) HPGDKLKB1CYP19A1CYP1A2SMN1; SMN2
SCHEMBL6071882 0.71 CYP19A1 (0.45) HPGDKLKB1CYP19A1CYP1A2SMN1; SMN2
SCHEMBL6071728 0.70 CYP19A1 (0.48) HPGDKLKB1CYP19A1CYP1A2SMN1; SMN2
SCHEMBL21467098 0.70 LMNA (0.48) LMNACA12CA1CA2CA3
SCHEMBL15924211 0.69 HPGD (0.60) HPGDKLKB1CYP19A1CYP1A2SMN1; SMN2
Trifluoroacetic Acid SCHEMBL8834496 0.67 CYP2C9 (0.41) HPGDKLKB1CYP19A1CYP1A2SMN1; SMN2
SCHEMBL795210 0.67 HPGD (0.68) HPGDKLKB1CYP19A1CYP1A2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014120783-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF NAUREX, INC. (US) 2014-08-07 WO disclosed