Acetic Acid

Acetic Acid

SCHEMBL15937484

CC(=O)O.N=C(N)c1nn(Cc2cncnc2)c2ncc(F)cc12

nearest known ligand 0.35

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA2AADRA2BADRA2CADRB2AGTR1AVPR1AAVPR1BAVPR2BDKRB2CALCRCHRNA3CHRNB4ESR1ESR2GHSRGNRHRGSC1HSPA8MALT1MC1RMC4RNOS1NOS2NOS3OPRK1OXTRRAMP1RAMP2RAMP3SCN5ASSTR1SSTR2SSTR3SSTR4SSTR5dacAdacBdacCfolPftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Acetic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 7/20 0.35
GRIN2B Q13224 7/20 0.35
GUCY1A1 Q02108 3/20 0.34
GUCY1B1 Q02153 3/20 0.34
PDE5A O76074 8/20 0.34
HDAC8 Q9BY41 1/20 0.32
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15937438 0.93 GRIN1 (0.34) GRIN1GRIN2BGUCY1A1GUCY1B1PDE5A
Acetic Acid SCHEMBL15937793 0.85 PDE5A (0.33) GUCY1A1GUCY1B1PDE5A
SCHEMBL19264469 0.84 GRIN1 (0.36) GRIN1GRIN2BPDE5A
Acetic Acid SCHEMBL15937721 0.84 GRIN1 (0.35) GRIN1GRIN2BGUCY1A1GUCY1B1PDE5A
Acetic Acid SCHEMBL15633156 0.84 PDE5A (0.48) GRIN1GRIN2BPDE5A
SCHEMBL14488217 0.82 GRIN1 (0.33) GRIN1GRIN2BPDE5A
SCHEMBL19244698 0.81 GRIN1 (0.34) GRIN1GRIN2BGUCY1A1GUCY1B1PDE5A
Acetic Acid SCHEMBL428284 0.81 PDE5A (0.48) GUCY1A1GUCY1B1PDE5A
Acetic Acid SCHEMBL16244961 0.81 PDE5A (0.34) GRIN1GRIN2BGUCY1A1GUCY1B1PDE5A
Acetic Acid SCHEMBL16244815 0.81 PTGDR2 (0.40) GUCY1A1GUCY1B1PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140228366-A1 HETEROARYL-SUBSTITUTED PYRAZOLOPYRIDINES AND USE THEREOF AS SOLUBLE GUANYLATE CYCLASE STIMULATORS BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-08-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140228366-A1 HETEROARYL-SUBSTITUTED PYRAZOLOPYRIDINES AND USE THEREOF AS SOLUBLE GUANYLATE CYCLASE STIMULATORS GUCY1A2, GUCY1B2, GUCY1B1 GRIN1 3030/4885GRIN2B 3045/4885GUCY1A1 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.