SCHEMBL15948985

SCHEMBL15948985

Cc1cc(C(=O)CC(c2cccc(-c3ccc(C(=O)O)c(F)c3)c2)c2ccccc2C)ccn1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.52
PSEN1 P49768 3/20 0.40
PSEN2 P49810 3/20 0.40
APH1B Q8WW43 3/20 0.40
NCSTN Q92542 3/20 0.40
APH1A Q96BI3 3/20 0.40
PSENEN Q9NZ42 3/20 0.40
CTSA P10619 10/20 0.39
NR3C2 P08235 1/20 0.38
S1PR1 P21453 1/20 0.37
S1PR3 Q99500 1/20 0.37
WNT3A P56704 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362685 0.93 GPBAR1 (0.61) GPBAR1PSEN1PSEN2APH1BNCSTN
SCHEMBL365553 0.91 GPBAR1 (0.47) GPBAR1PSEN1PSEN2APH1BNCSTN
SCHEMBL1389580 0.90 GPBAR1 (0.68) GPBAR1PSEN1PSEN2APH1BNCSTN
SCHEMBL364591 0.90 GPBAR1 (0.68) GPBAR1PSEN1PSEN2APH1BNCSTN
SCHEMBL364000 0.87 GPBAR1 (0.57) GPBAR1PSEN1PSEN2APH1BNCSTN
SCHEMBL362655 0.85 GPBAR1 (0.61) GPBAR1PSEN1PSEN2APH1BNCSTN
SCHEMBL362597 0.85 GPBAR1 (0.54) GPBAR1PSEN1PSEN2APH1BNCSTN
SCHEMBL369861 0.84 GPBAR1 (0.55) GPBAR1PSEN1PSEN2APH1BNCSTN
SCHEMBL10291336 0.84 GPBAR1 (0.59) GPBAR1PSEN1PSEN2APH1BNCSTN
SCHEMBL371338 0.83 GPBAR1 (0.55) GPBAR1PSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-B1 1-HYDROXYIMINO-3-PHENYL-PROPANES HOFFMANN LA ROCHE (CH) 2014-08-20 EP disclosed