SCHEMBL15949047

SCHEMBL15949047

O=C(O)Oc1ccc(-c2ccc(C(C/C(=N\O)c3ccncc3)c3ccccc3)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 3/20 0.59
EPHX2 P34913 1/20 0.39
FFAR1 O14842 3/20 0.39
GSK3B P49841 5/20 0.39
ROCK1 Q13464 5/20 0.39
CLK4 Q9HAZ1 5/20 0.39
RPS6KA5 O75582 4/20 0.39
AKT1 P31749 4/20 0.39
PRKCD Q05655 4/20 0.39
PRKG2 Q13237 4/20 0.39
PRKG1 Q13976 4/20 0.39
PKN2 Q16513 4/20 0.39
GSK3A P49840 4/20 0.39
NEK4 P51957 3/20 0.39
ROCK2 O75116 3/20 0.39
MAP4K4 O95819 3/20 0.39
CDK1 P06493 3/20 0.39
RPS6KB1 P23443 3/20 0.39
CDK2 P24941 3/20 0.39
MAPK1 P28482 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15949238 0.90 GPBAR1 (0.54) GPBAR1FFAR1GSK3BROCK1CLK4
SCHEMBL363119 0.85 GPBAR1 (0.64) GPBAR1EPHX2GSK3BROCK1CLK4
SCHEMBL1389878 0.85 GPBAR1 (0.64) GPBAR1EPHX2GSK3BROCK1CLK4
SCHEMBL1390378 0.83 GPBAR1 (0.61) GPBAR1EPHX2GSK3BROCK1CLK4
SCHEMBL1390380 0.83 GPBAR1 (0.61) GPBAR1EPHX2GSK3BROCK1CLK4
SCHEMBL363952 0.82 GPBAR1 (0.76) GPBAR1EPHX2MEN1KMT2ALMNA
SCHEMBL368449 0.82 GPBAR1 (0.76) GPBAR1EPHX2MEN1KMT2ALMNA
SCHEMBL368448 0.82 GPBAR1 (0.76) GPBAR1EPHX2MEN1KMT2ALMNA
SCHEMBL1390074 0.81 GPBAR1 (0.64) GPBAR1EPHX2GSK3BROCK1CLK4
SCHEMBL369535 0.81 GPBAR1 (0.64) GPBAR1EPHX2GSK3BROCK1CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-B1 1-HYDROXYIMINO-3-PHENYL-PROPANES HOFFMANN LA ROCHE (CH) 2014-08-20 EP claimed