SCHEMBL15949320

SCHEMBL15949320

Cc1cc(/C(C[C@H](c2ccc(N3C[C@@H]4C(OC(=O)O)[C@@H]4C3)cc2)c2ccc(F)cc2F)=N/O)ccn1

nearest known ligand 0.64

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 4/20 0.64
ACACB O00763 3/20 0.32
KEAP1 Q14145 2/20 0.32
NFE2L2 Q16236 2/20 0.32
KDM5A P29375 1/20 0.31
KDM4C Q9H3R0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1390002 0.90 GPBAR1 (0.76) GPBAR1ACACBKEAP1NFE2L2KDM5A
SCHEMBL1390399 0.90 GPBAR1 (0.76) GPBAR1ACACBKEAP1NFE2L2KDM5A
SCHEMBL1390400 0.90 GPBAR1 (0.76) GPBAR1ACACBKEAP1NFE2L2KDM5A
SCHEMBL1390006 0.90 GPBAR1 (0.76) GPBAR1ACACBKEAP1NFE2L2KDM5A
SCHEMBL1390005 0.90 GPBAR1 (0.76) GPBAR1ACACBKEAP1NFE2L2KDM5A
SCHEMBL15949197 0.88 GPBAR1 (0.65) GPBAR1ACACBKDM5AKDM4C
SCHEMBL15949262 0.88 GPBAR1 (0.65) GPBAR1ACACBKDM5AKDM4C
SCHEMBL1390449 0.88 GPBAR1 (0.64) GPBAR1ACACBKEAP1NFE2L2KDM5A
SCHEMBL1390448 0.88 GPBAR1 (0.64) GPBAR1ACACBKEAP1NFE2L2KDM5A
SCHEMBL1389807 0.83 GPBAR1 (0.69) GPBAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-B1 1-HYDROXYIMINO-3-PHENYL-PROPANES HOFFMANN LA ROCHE (CH) 2014-08-20 EP claimed