SCHEMBL1595880

SCHEMBL1595880

CO[C@@H](c1ccc(C(F)(F)F)cc1)[C@@H](CO)N(C(=O)O)C(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.39
AKR1C2 P52895 2/20 0.39
FFAR1 O14842 5/20 0.36
EEF2K O00418 1/20 0.35
MEN1 O00255 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
ALOX15 P16050 1/20 0.35
SLC6A1 P30531 1/20 0.35
KMT2A Q03164 1/20 0.35
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35
CNR2 P34972 1/20 0.34
SLC6A9 P48067 1/20 0.34
LDHA P00338 1/20 0.34
LDHB P07195 1/20 0.34
PPARG P37231 2/20 0.34
PPARD Q03181 1/20 0.34
PPARA Q07869 1/20 0.34
UTS2R Q9UKP6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1596367 0.85 AKR1C3 (0.33) AKR1C3AKR1C2FFAR1EEF2KMEN1
SCHEMBL1595011 0.83 AKR1C3 (0.40) AKR1C3AKR1C2FFAR1EEF2KCES2
SCHEMBL2548060 0.83 AKR1C3 (0.37) AKR1C3AKR1C2FFAR1MEN1CYP3A4
SCHEMBL1595216 0.83 AKR1C3 (0.37) AKR1C3AKR1C2FFAR1MEN1CYP3A4
SCHEMBL1742949 0.79 CES2 (0.37) AKR1C3AKR1C2FFAR1EEF2KCES2
SCHEMBL1742950 0.79 CES2 (0.37) AKR1C3AKR1C2FFAR1EEF2KCES2
SCHEMBL2544467 0.79 CES2 (0.37) AKR1C3AKR1C2FFAR1EEF2KCES2
SCHEMBL1594812 0.79 SLC6A4 (0.39) AKR1C3AKR1C2FFAR1EEF2KCYP3A4
SCHEMBL2549587 0.78 FFAR1 (0.34) AKR1C3AKR1C2FFAR1EEF2KCES2
SCHEMBL1594707 0.78 FFAR1 (0.34) AKR1C3AKR1C2FFAR1EEF2KCES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7919504-B2 Thiadiazole modulators of PKB AMGEN INC. (US) 2011-04-05 US disclosed