SCHEMBL15959068

SCHEMBL15959068

Bc1ccc([C@@H](C)N2CCC(CC=C)(c3ccccc3)OC2=O)cc1

nearest known ligand 0.57

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 18/20 0.57
CYP2C9 P11712 14/20 0.57
CYP3A4 P08684 11/20 0.57
CYP2C19 P33261 9/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1755289 1.00 HSD11B1 (0.57) HSD11B1CYP2C9CYP3A4CYP2C19
SCHEMBL1755333 1.00 HSD11B1 (0.57) HSD11B1CYP2C9CYP3A4CYP2C19
SCHEMBL958708 0.92 HSD11B1 (0.57) HSD11B1CYP2C9CYP3A4CYP2C19
SCHEMBL1755291 0.92 HSD11B1 (0.57) HSD11B1CYP2C9CYP3A4CYP2C19
SCHEMBL958709 0.92 HSD11B1 (0.57) HSD11B1CYP2C9CYP3A4CYP2C19
SCHEMBL956672 0.91 HSD11B1 (0.70) HSD11B1CYP2C9CYP3A4CYP2C19
SCHEMBL736173 0.91 HSD11B1 (0.70) HSD11B1CYP2C9CYP3A4CYP2C19
SCHEMBL956702 0.91 HSD11B1 (0.69) HSD11B1CYP2C9CYP3A4CYP2C19
SCHEMBL117313 0.91 HSD11B1 (0.70) HSD11B1CYP2C9CYP3A4CYP2C19
SCHEMBL959511 0.91 HSD11B1 (0.56) HSD11B1CYP2C9CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2183228-B1 CYCLIC INHIBITORS OF 11ß -HYDROXYSTERIOD DEHYDROGENASE 1 VITAE PHARMACEUTICALS INC (US) 2014-08-20 EP disclosed