SCHEMBL15961237

SCHEMBL15961237

CN1C(=O)C[C@]2(CCc3ccc([N+](=O)[O-])cc32)N=C1NC(=O)O

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.35
WDR5 P61964 5/20 0.34
ALDH1A1 P00352 3/20 0.34
LMNA P02545 2/20 0.34
POLB P06746 2/20 0.34
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
TAS1R2 Q8TE23 1/20 0.34
KMT2A Q03164 1/20 0.34
GAA P10253 1/20 0.34
RXRA P19793 1/20 0.33
RXRB P28702 1/20 0.33
RXRG P48443 1/20 0.33
NR3C1 P04150 1/20 0.33
PTGES O14684 1/20 0.33
MAPT P10636 1/20 0.33
HSPA9 P38646 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15961238 1.00 SIRT2 (0.35) SIRT2WDR5ALDH1A1LMNAPOLB
SCHEMBL15976459 0.87 BACE1 (0.47) SIRT2ALDH1A1LMNAMAPT
SCHEMBL10198037 0.84 LMNA (0.38) SIRT2ALDH1A1LMNAPOLBKMT2A
SCHEMBL2892930 0.83 BACE1 (0.35)
SCHEMBL568438 0.81 LMNA (0.33) SIRT2ALDH1A1LMNAKMT2AGAA
SCHEMBL8516276 0.67 BACE2 (0.41) WDR5KMT2AMAPT
SCHEMBL8516273 0.67 BACE2 (0.41) WDR5KMT2AMAPT
SCHEMBL8516270 0.67 BACE2 (0.41) WDR5KMT2AMAPT
SCHEMBL299015 0.67 BACE1 (0.44) WDR5ALDH1A1GAAMAPT
SCHEMBL299014 0.67 BACE1 (0.44) WDR5ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8815881-B2 1,4,5,6-tetrahydro-pyrimidin-2-ylamine compounds HOFFMANN-LA ROCHE INC. (US) 2014-08-26 US disclosed