SCHEMBL15975833

SCHEMBL15975833

Cc1ncc(-c2cnc3sc(-c4ccc5c(c4)C4(CCNCC4)C(=O)N5)nn23)cc1C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 13/20 0.48
PGR P06401 2/20 0.35
ALPL P05186 1/20 0.34
ALPI P09923 1/20 0.34
PIK3CD O00329 2/20 0.34
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
NPC1 O15118 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL531960 0.90 PIK3CA (0.56) PIK3CAPGR
SCHEMBL2124315 0.78 PIK3CA (0.53) PIK3CAPIK3CD
SCHEMBL2122854 0.77 PIK3CA (0.42) PIK3CAPIK3CD
SCHEMBL15975840 0.75 PIK3CA (0.47) PIK3CAPIK3CD
SCHEMBL15975832 0.73 PIK3CA (0.59) PIK3CA
SCHEMBL15975827 0.72 PIK3CA (0.79) PIK3CA
SCHEMBL15975838 0.71 PIK3CA (0.55) PIK3CAALPLALPI
SCHEMBL15975837 0.70 PIK3CA (0.63) PIK3CA
SCHEMBL532219 0.68 PIK3CA (0.82) PIK3CA
SCHEMBL15975830 0.68 PIK3CA (0.68) PIK3CAMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8815918-B2 Imidazo [2, 1-B] [1, 3, 4] thiadiazole derivatives CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO) (ES) 2014-08-26 US disclosed