SCHEMBL15977152

SCHEMBL15977152

Fc1c(F)c(F)c(Nc2nc(-c3cccnc3)nc3ccccc23)c(F)c1F

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 5/20 0.75
CYP3A4 P08684 5/20 0.75
TSHR P16473 4/20 0.75
CYP2C19 P33261 4/20 0.75
HSD17B10 Q99714 4/20 0.75
MAPK1 P28482 4/20 0.75
MAPT P10636 3/20 0.75
KDM4E B2RXH2 2/20 0.75
HPGD P15428 2/20 0.75
TDP1 Q9NUW8 1/20 0.75
CLK4 Q9HAZ1 4/20 0.72
ALDH1A1 P00352 4/20 0.72
LMNA P02545 3/20 0.72
USP2 O75604 2/20 0.72
ABCG2 Q9UNQ0 3/20 0.69
CYP2D6 P10635 3/20 0.66
CYP2C9 P11712 1/20 0.66
POLB P06746 1/20 0.65
HTT P42858 1/20 0.65
PDE5A O76074 3/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL15966651 0.99 CYP1A2 (0.73) CYP1A2CYP3A4TSHRCYP2C19HSD17B10
SCHEMBL15977150 0.84 CYP1A2 (0.67) CYP1A2CYP3A4TSHRCYP2C19HSD17B10
SCHEMBL15986596 0.84 CYP1A2 (0.78) CYP1A2CYP3A4TSHRCYP2C19HSD17B10
SCHEMBL7280796 0.84 CYP1A2 (1.00) CYP1A2CYP3A4TSHRCYP2C19HSD17B10
Hydrochloric Acid SCHEMBL15966802 0.83 CYP1A2 (0.66) CYP1A2CYP3A4TSHRCYP2C19HSD17B10
Hydrochloric Acid SCHEMBL15966650 0.83 CYP1A2 (0.76) CYP1A2CYP3A4TSHRCYP2C19HSD17B10
SCHEMBL1083757 0.81 MAPT (0.80) CYP1A2CYP3A4TSHRCYP2C19HSD17B10
SCHEMBL20273653 0.80 CYP1A2 (1.00) CYP1A2CYP3A4TSHRCYP2C19HSD17B10
SCHEMBL15977138 0.79 CYP1A2 (0.66) CYP1A2CYP3A4TSHRCYP2C19HSD17B10
SCHEMBL1062324 0.79 PDE5A (1.00) CYP1A2CYP3A4TSHRCYP2C19HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014128206-A1 COMPOUNDS FOR USE IN INHIBITING HIV CAPSID ASSEMBLY Ruprecht-Karls-Universität Heidelberg (DE) 2014-08-28 WO disclosed
EP-2769723-A1 Compounds for use in inhibiting HIV capsid assembly Ruprecht-Karls-Universität Heidelberg (DE) 2014-08-27 EP disclosed