SCHEMBL15977155

SCHEMBL15977155

CN(C)c1nc(-c2cccnc2)nc2ccc(O)cc12

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.70
CYP3A4 P08684 2/20 0.70
CYP2D6 P10635 2/20 0.70
CYP2C9 P11712 2/20 0.70
CLK4 Q9HAZ1 2/20 0.70
MEN1 O00255 2/20 0.70
KMT2A Q03164 2/20 0.70
ALDH1A1 P00352 1/20 0.70
GLA P06280 1/20 0.70
TSHR P16473 1/20 0.70
GBA1 P04062 15/20 0.53
LMNA P02545 1/20 0.50
MAPK1 P28482 1/20 0.50
HIF1A Q16665 1/20 0.50
RXFP1 Q9HBX9 1/20 0.50
LATS1 O95835 1/20 0.50
LATS2 Q9NRM7 1/20 0.50
KDM4E B2RXH2 1/20 0.49
POLB P06746 1/20 0.49
GAA P10253 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL15966750 0.99 CYP1A2 (0.68) CYP1A2CYP3A4CYP2D6CYP2C9CLK4
SCHEMBL16183452 0.90 CYP1A2 (0.64) CYP1A2CYP3A4CYP2D6CYP2C9CLK4
SCHEMBL14727523 0.85 CYP1A2 (0.70) CYP1A2CYP3A4CYP2D6CYP2C9CLK4
SCHEMBL20609337 0.82 ALDH1A1 (1.00) CYP1A2CYP3A4CYP2D6CYP2C9CLK4
SCHEMBL14474975 0.81 MEN1 (0.65) CYP1A2CYP3A4CYP2D6CYP2C9CLK4
SCHEMBL14475027 0.81 CYP1A2 (0.65) CYP1A2CYP3A4CYP2D6CYP2C9CLK4
SCHEMBL14475090 0.81 CYP1A2 (0.65) CYP1A2CYP3A4CYP2D6CYP2C9CLK4
SCHEMBL14475135 0.81 CYP3A4 (0.61) CYP1A2CYP3A4CYP2D6CYP2C9CLK4
SCHEMBL14475059 0.81 CYP1A2 (0.61) CYP1A2CYP3A4CYP2D6CYP2C9CLK4
SCHEMBL14475208 0.81 CYP1A2 (0.64) CYP1A2CYP3A4CYP2D6CYP2C9CLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014128206-A1 COMPOUNDS FOR USE IN INHIBITING HIV CAPSID ASSEMBLY Ruprecht-Karls-Universität Heidelberg (DE) 2014-08-28 WO disclosed
EP-2769723-A1 Compounds for use in inhibiting HIV capsid assembly Ruprecht-Karls-Universität Heidelberg (DE) 2014-08-27 EP disclosed