SCHEMBL15980908

SCHEMBL15980908

Cc1ccc(-c2c(C)noc2C)cc1S(C)(=O)=O

nearest known ligand 0.76

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 20/20 0.76
BRD2 P25440 17/20 0.76
BRD3 Q15059 17/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14740758 0.87 BRD4 (1.00) BRD4BRD2BRD3
SCHEMBL14740769 0.87 BRD4 (0.74) BRD4BRD2BRD3
SCHEMBL15980898 0.85 BRD4 (0.72) BRD4BRD2BRD3
SCHEMBL15980799 0.84 BRD4 (0.76) BRD4BRD2BRD3
SCHEMBL14756139 0.81 BRD4 (0.71) BRD4BRD2BRD3
SCHEMBL14756377 0.79 BRD4 (0.85) BRD4BRD2BRD3
SCHEMBL14756381 0.79 BRD4 (0.85) BRD4BRD2BRD3
SCHEMBL15984849 0.79 BRD4 (1.00) BRD4BRD2BRD3
SCHEMBL15782904 0.79 BRD4 (0.62) BRD4BRD2BRD3
SCHEMBL12338501 0.78 BRD4 (0.63) BRD4BRD2BRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140243286-A1 BROMODOMAIN LIGANDS CAPABLE OF DIMERIZING IN AN AQUEOUS SOLUTION, AND METHODS OF USING SAME COFERON, INC. (US) 2014-08-28 US disclosed
US-20140243322-A1 BIVALENT BROMODOMAIN LIGANDS, AND METHODS OF USING SAME COFERON, INC. (US) 2014-08-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140243322-A1 BIVALENT BROMODOMAIN LIGANDS, AND METHODS OF USING SAME BRDT, BRD2, BRD4 BRD4 3/4885BRD2 2/4885BRD3 4/4885
US-20140243286-A1 BROMODOMAIN LIGANDS CAPABLE OF DIMERIZING IN AN AQUEOUS SOLUTION, AND METHODS OF USING SAME BRDT, BRD4, BRD1 BRD4 2/4885BRD2 5/4885BRD3 6/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.