Zacopride

Zacopride

SCHEMBL16003

COc1cc(N)c(Cl)cc1C(=O)NC1CN2CCC1CC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 4/20 1.00
HTR3E A5X5Y0 2/20 1.00
HTR3B O95264 2/20 1.00
HTR3D Q70Z44 2/20 1.00
HTR3C Q8WXA8 2/20 1.00
HTR5A P47898 1/20 1.00
MEN1 O00255 1/20 1.00
CYP2D6 P10635 1/20 1.00
CYP2C9 P11712 1/20 1.00
CYP2C19 P33261 1/20 1.00
KMT2A Q03164 1/20 1.00
MAPK1 P28482 1/20 0.96
NPSR1 Q6W5P4 1/20 0.77
ADRA2A P08913 1/20 0.62
ADRA2B P18089 1/20 0.62
ADRA2C P18825 1/20 0.62
HTR2A P28223 1/20 0.62
HTR2C P28335 1/20 0.62
HTR2B P41595 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
(R)Zacopride SCHEMBL5387843 1.00 HTR3A (1.00) HTR3AHTR3EHTR3BHTR3DHTR3C
Zacopride SCHEMBL5373467 1.00 HTR3A (1.00) HTR3AHTR3EHTR3BHTR3DHTR3C
Zacopride SCHEMBL29567897 1.00 HTR3A (1.00) HTR3AHTR3EHTR3BHTR3DHTR3C
Zacopride SCHEMBL7280998 0.99 MAPK1 (0.98) HTR3AHTR3EHTR3BHTR3DHTR3C
Zacopride SCHEMBL7281576 0.99 MAPK1 (0.98) HTR3AHTR3EHTR3BHTR3DHTR3C
Zacopride SCHEMBL667580 0.99 MAPK1 (0.98) HTR3AHTR3EHTR3BHTR3DHTR3C
Zacopride SCHEMBL7280994 0.99 MAPK1 (0.98) HTR3AHTR3EHTR3BHTR3DHTR3C
Zacopride SCHEMBL9598323 0.98 MAPK1 (1.00) HTR3AHTR3EHTR3BHTR3DHTR3C
Zacopride SCHEMBL29389976 0.98 MAPK1 (1.00) HTR3AHTR3EHTR3BHTR3DHTR3C
Zacopride SCHEMBL7288008 0.94 HTR3A (0.88) HTR3AHTR3EHTR3BHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2032 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116211847-A Application of saururus chinensis ketone in preparation of medicine for preventing and/or treating irritable bowel syndrome 四川省医学科学院·四川省人民医院 2023-06-06 CN claimed
US-11571397-B2 Compositions and methods for treating seizure-induced sudden death ZOGENIX INTERNATIONAL LIMITED (GB) 2023-02-07 US claimed
US-20220313686-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING A COMBINATION OF OPIOID ANTAGONISTS YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM LTD. (IL) 2022-10-06 US claimed
US-20220273680-A1 Methods of Treating Psychological and Brain Disorders UNIVERSITY OF MARYLAND, BALTIMORE (US) 2022-09-01 US claimed
EP-4013403-A1 METHODS OF TREATING PSYCHOLOGICAL AND BRAIN DISORDERS University of Maryland, Baltimore (US) 2022-06-22 EP claimed
EP-4013390-A1 PHARMACEUTICAL COMPOSITIONS COMPRISING A COMBINATION OF OPIOID ANTAGONISTS YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM LTD (IL) 2022-06-22 EP claimed
CN-114599355-A Method for treating psychological and cerebral diseases 马里兰大学巴尔的摩分校 2022-06-07 CN claimed
US-20220146492-A1 CELL MEMBRANE PERMEABILITY RESTORING THERAPY SHINE IAN BASIL (US) 2022-05-12 US claimed
EP-3953000-A1 CELL MEMBRANE PERMEABILITY RESTORING THERAPY Shine, Ian Basil (US) 2022-02-16 EP claimed
US-20210338647-A1 Combination of Acetylcholinesterase Inhibitor and 5-HT4 Receptor Agonist As Neuroprotective Agent In the Treatment of Neurodegenerative Diseases CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2021-11-04 US claimed
EP-0327335-A1 Arylamido(and arylthioamido)-azabicycloalkanes for enhancing memory or correcting memory deficiency SYNTHELABO (FR) 1989-08-09 EP claimed
EP-0311724-A1 Anxiolytic-R-N-(1-azabicyclo[2.2.2]oct-3-yl) benzamides and thiobenzamides SYNTHELABO (FR) 1989-04-19 EP claimed
EP-0306345-A2 2-Alkoxy-n-(1-azabicyclo(2.2.2)-oct-3-yl) benzamides and thiobenzamides having an antischizophrenic activity SYNTHELABO (FR) 1989-03-08 EP claimed
EP-0272052-A1 Anxiolytic-N-(1-Azabicyclo[2.2.2]Oct-3-yl) Benzamides and Thobenzamides A.H. ROBINS COMPANY, INCORPORATED (a Delaware corporation) (US) 1988-06-22 EP claimed
US-4717563-A 2-alkoxy-N-(1-azabicyclo(2.2.2)oct-3-yl) benzamides and thiobenzamides in a method for alleviating emesis caused by non-platinum anticancer drugs A. H. ROBINS COMPANY, INC. (US) 1988-01-05 US claimed
EP-0240180-A1 2-alkoxy-N-(1-azabicyclo[2.2.2]-oct-3-yl) benzamides and thiobenzamides in the alleviation of emesis caused by non-platinum anticancer drugs SYNTHELABO (FR) 1987-10-07 EP claimed
EP-0190920-A2 Method of enhancing memory or correcting memory deficiency with arylamido (and arylthioamido)azabicycloalkanes SYNTHELABO (FR) 1986-08-13 EP claimed
US-4605652-A ALZHEIMER'S DISEASE; SENILITY A. H. ROBINS COMPANY, INC. (US) 1986-08-12 US claimed
US-4593034-A 2-alkoxy-N-(1-azabicyclo[2.2.2]oct-3-yl)benzamides and thiobenzamides A. H. ROBINS COMPANY, INC. (US) 1986-06-03 US claimed
EP-0158532-A2 Use of 4-amino-N-(1-azabicyclo[2.2.2]oct-3-yl)-5-chloro-2-methoxybenzamide for the manufacture of a medicament having anti-emetic activity. SYNTHELABO (FR) 1985-10-16 EP claimed