SCHEMBL16004452

SCHEMBL16004452

CC1c2cc(C=O)ccc2OCCN1C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 2/20 0.38
GHSR Q92847 1/20 0.37
ATM Q13315 2/20 0.36
SCD5 Q86SK9 1/20 0.35
GPR119 Q8TDV5 2/20 0.35
ALDH1A1 P00352 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
OPRK1 P41145 1/20 0.33
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
HPGD P15428 1/20 0.33
RAB9A P51151 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CSNK2A2 P19784 1/20 0.33
CSNK2A1 P68400 1/20 0.33
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29501163 0.84 HCRTR2 (0.43) USP30ATMSCD5GPR119MEN1
SCHEMBL17958021 0.84 HCRTR2 (0.43) USP30ATMSCD5GPR119MEN1
SCHEMBL30878572 0.81 GHSR (0.46) GHSRNPC1RAB9AKMT2ALMNA
SCHEMBL5776208 0.81 GHSR (0.46) GHSRNPC1RAB9AKMT2ALMNA
SCHEMBL17973702 0.79 DRD3 (0.41) ATMALDH1A1KDM4ENPC1HPGD
SCHEMBL17973703 0.79 DRD3 (0.41) ATMALDH1A1KDM4ENPC1HPGD
SCHEMBL18616603 0.78 GHSR (0.50) GHSRNR1H2
SCHEMBL2878054 0.78 EGFR (0.45) USP30ALDH1A1HSD17B10TDP1KMT2A
SCHEMBL30418523 0.78 EGFR (0.45) USP30ALDH1A1HSD17B10TDP1KMT2A
SCHEMBL17958028 0.77 USP30 (0.40) USP30ATMSCD5MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014133414-A2 HETEROCYCLIC TGR5 BILE ACID RECEPTOR AGONISTS, PHARMACEUTICAL COMPOSITION, METHODS FOR THE PRODUCTION AND USE THEREOF АЛЛА ХЕМ ЛЛС (US) 2014-09-04 WO disclosed