SCHEMBL16011997

SCHEMBL16011997

NC(N)=Nc1cccc(-c2ccnc3[nH]c4ccccc4c23)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.43
PTK6 Q13882 6/20 0.43
ALK Q9UM73 5/20 0.43
ERBB2 P04626 4/20 0.43
AURKA O14965 1/20 0.43
EGFR P00533 1/20 0.43
SRC P12931 1/20 0.43
ACVR1 Q04771 1/20 0.43
AURKC Q9UQB9 1/20 0.43
PLG P00747 1/20 0.42
NUDT1 P36639 1/20 0.39
PRKCI P41743 1/20 0.39
PLAU P00749 2/20 0.38
HTR3E A5X5Y0 1/20 0.38
SLC22A2 O15244 1/20 0.38
SLC22A1 O15245 1/20 0.38
SLC22A3 O75751 1/20 0.38
HTR3B O95264 1/20 0.38
HTR3A P46098 1/20 0.38
HTR3D Q70Z44 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16011816 0.81 GRIN2D (0.43) MAPK14PTK6ALKERBB2AURKA
SCHEMBL16024047 0.80 ERBB2 (0.61) MAPK14PTK6ALKERBB2AURKA
SCHEMBL16011993 0.80 MAPK14 (0.48) MAPK14PTK6ALKERBB2AURKA
SCHEMBL16011996 0.78 PTK6 (0.47) MAPK14PTK6ALKERBB2AURKA
SCHEMBL17471213 0.78 PTK6 (0.49) MAPK14PTK6ALKERBB2AURKA
SCHEMBL16257469 0.77 LRRK2 (0.53) MAPK14PTK6ALKERBB2AURKA
SCHEMBL16011810 0.77 EGFR (0.47) MAPK14PTK6ALKERBB2AURKA
SCHEMBL16011815 0.76 F3 (0.42) MAPK14PTK6ALKERBB2AURKA
SCHEMBL23967926 0.75 PTK6 (0.49) MAPK14PTK6ALKERBB2AURKA
SCHEMBL674288 0.75 MAPK14 (0.60) MAPK14PTK6ALKERBB2ACVR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2964225-A1 CaMKII INHIBITORS AND USES THEREOF Allosteros Therapeutics Inc. (US) 2016-01-13 EP disclosed
WO-2014138212-A1 CaMKII INHIBITORS AND USES THEREOF ALLOSTEROS THERAPEUTICS, INC. (US) 2014-09-12 WO disclosed