SCHEMBL16014124

SCHEMBL16014124

NC(Cc1ccccc1)c1cccc2[nH]ccc12

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.46
DRD4 P21917 3/20 0.44
DRD3 P35462 3/20 0.44
DRD2 P14416 2/20 0.44
HPGDS O60760 1/20 0.43
SLC6A2 P23975 2/20 0.42
TAAR1 Q96RJ0 2/20 0.42
MAOA P21397 1/20 0.42
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
CYP2A6 P11509 1/20 0.42
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
IDO1 P14902 1/20 0.41
EPHX1 P07099 1/20 0.40
AHR P35869 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27556122 0.80 AHR (0.48) CYP19A1DRD4DRD3SLC6A3AHR
SCHEMBL29816334 0.79 AHR (0.43) CYP19A1AHR
SCHEMBL6563314 0.77 MCL1 (0.40) HPGDSAHR
SCHEMBL3283005 0.75 ACP3 (0.55) SLC6A2TAAR1MAOASLC6A4SLC6A3
SCHEMBL16014125 0.74 MEN1 (0.52) SLC6A2TAAR1SLC6A4AHR
SCHEMBL23432526 0.73 AHR (0.47) CYP19A1DRD4DRD3SLC6A3AHR
SCHEMBL3730120 0.73 AHR (0.47) SLC6A2SLC6A4SLC6A3AHR
SCHEMBL10502553 0.72 GPR84 (0.57) SLC6A2SLC6A4AHR
SCHEMBL3095729 0.72 HRH1 (0.52) HPGDSSLC6A2SLC6A4AHR
SCHEMBL27721184 0.71 CYP2D6 (0.42) DRD4DRD3DRD2HPGDSSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2964225-A1 CaMKII INHIBITORS AND USES THEREOF Allosteros Therapeutics Inc. (US) 2016-01-13 EP disclosed
WO-2014138212-A1 CaMKII INHIBITORS AND USES THEREOF ALLOSTEROS THERAPEUTICS, INC. (US) 2014-09-12 WO disclosed