SCHEMBL16024596

SCHEMBL16024596

C=CC(C)(C)c1ccc2c(c1)OCCN(Cc1ccc(OC)cc1)C2=O

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TNIK Q9UKE5 12/20 0.53
ROCK2 O75116 7/20 0.52
ROCK1 Q13464 5/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16014462 0.92 TNIK (0.54) TNIKROCK2ROCK1
SCHEMBL16014355 0.80 TNIK (0.58) TNIKROCK2ROCK1
SCHEMBL17957873 0.77 ROCK2 (0.60) TNIKROCK2ROCK1
SCHEMBL17368202 0.76 ROCK2 (0.45) TNIKROCK2ROCK1
SCHEMBL17957628 0.75 TNIK (0.56) TNIKROCK2ROCK1
SCHEMBL1726059 0.74 GAA (0.46) TNIKROCK2ROCK1
SCHEMBL8365726 0.72 GAA (0.50) TNIKROCK2ROCK1
SCHEMBL17957654 0.71 ROCK2 (0.53) TNIKROCK2ROCK1
SCHEMBL19929676 0.70 ROCK2 (0.72) TNIKROCK2ROCK1
SCHEMBL28882904 0.69 ROCK2 (0.71) TNIKROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2964642-B1 INHIBITORS OF BRUTON'S TYROSINE KINASE HOFFMANN LA ROCHE (CH) 2017-11-15 EP disclosed
WO-2014135474-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE F. HOFFMANN-LA ROCHE AG (CH) 2014-09-12 WO disclosed