SCHEMBL16038147

SCHEMBL16038147

Cc1nc([N+](=O)[O-])ccc1Oc1ccnc(NC(=O)N2CCCC2)c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 9/20 0.44
PDGFRA P16234 6/20 0.44
KIT P10721 3/20 0.44
PDGFRB P09619 2/20 0.43
AXL P30530 2/20 0.42
TGFBR1 P36897 5/20 0.42
MET P08581 3/20 0.42
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GLA P06280 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
KLK7 P49862 1/20 0.40
RAB9A P51151 1/20 0.40
CYP2C9 P11712 1/20 0.39
PIK3C3 Q8NEB9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30890878 0.93 CSF1R (0.45) CSF1RPDGFRAKITPDGFRBTGFBR1
SCHEMBL16036512 0.93 CSF1R (0.45) CSF1RPDGFRAKITPDGFRBTGFBR1
SCHEMBL16036505 0.86 TGFBR1 (0.45) CSF1RPDGFRAKITPDGFRBTGFBR1
SCHEMBL16036508 0.86 TGFBR1 (0.45) CSF1RPDGFRAKITPDGFRBTGFBR1
SCHEMBL16038009 0.85 CSF1R (0.52) CSF1RPDGFRAPDGFRBTGFBR1MET
SCHEMBL16037333 0.84 CSF1R (0.45) CSF1RPDGFRAKITPDGFRBAXL
SCHEMBL13860835 0.83 GAA (0.46) AXLMETALDH1A1GAA
SCHEMBL16038204 0.83 KDR (0.49)
SCHEMBL21772037 0.83 KDR (0.51) CSF1RPDGFRAPDGFRB
SCHEMBL16037125 0.82 TGFBR1 (0.43) CSF1RPDGFRAKITPDGFRBAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9309224-B2 N-acyl-N′-(pyridin-2-yl) ureas and analogs exhibiting anti-cancer and anti-proliferative activities DECIPHERA PHARMACEUTICALS, LLC. (US) 2016-04-12 US disclosed
US-20140275016-A1 N-Acyl-N'-(pyridin-2-yl) Ureas and Analogs Exhibiting Anti-Cancer and Anti-Proliferative Activities DECIPHERA PHARMACEUTICALS, LLC (US) 2014-09-18 US disclosed
WO-2014145029-A2 N-ACYL-N'-(PYRIDIN-2-YL) UREAS AND ANALOGS EXHIBITING ANTI-CANCER AND ANTI-PROLIFERATIVE ACTIVITIES DECIPHERA PHARMACEUTICALS, LLC (US) 2014-09-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140275016-A1 N-Acyl-N'-(pyridin-2-yl) Ureas and Analogs Exhibiting Anti-Cancer and Anti-Proliferative Activities KIT, CSF1R, CSF3R CSF1R 2/4885PDGFRA 5/4885KIT 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.