SCHEMBL16059774

SCHEMBL16059774

Cc1noc(C)c1-c1ccc2[nH]ccc2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 13/20 1.00
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
RAB9A P51151 1/20 0.60
LMNA P02545 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
CREBBP Q92793 2/20 0.56
JAK2 O60674 1/20 0.55
BRD2 P25440 3/20 0.47
NPC1 O15118 1/20 0.46
BRD3 Q15059 1/20 0.46
ERN1 O75460 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31735610 1.00 BRD4 (1.00) BRD4MEN1KMT2ARAB9ALMNA
SCHEMBL18124120 0.88 BRD4 (1.00) BRD4MEN1KMT2ARAB9ALMNA
SCHEMBL31735700 0.88 BRD4 (1.00) BRD4MEN1KMT2ARAB9ALMNA
SCHEMBL17581483 0.78 BRD4 (0.63) BRD4CREBBPJAK2BRD2
SCHEMBL29422776 0.77 BRD4 (0.64) BRD4CREBBP
SCHEMBL859173 0.77 BRD4 (0.64) BRD4CREBBP
SCHEMBL31735707 0.76 BRD4 (0.65) BRD4CREBBPJAK2BRD2BRD3
SCHEMBL19998616 0.76 BRD4 (0.65) BRD4CREBBPJAK2BRD2BRD3
SCHEMBL24717312 0.75 BRD4 (0.60) BRD4CREBBPJAK2BRD2BRD3
SCHEMBL24913618 0.75 BRD4 (0.79) BRD4LMNACREBBPJAK2BRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025245484-A1 FOXN1 ACTIVATORS THYMOFOX INC. (US) 2025-11-27 WO disclosed
EP-2970265-B1 HETEROCYCLIC COMPOUNDS AND USES THEREOF PLEXXIKON INC (US) 2018-08-08 EP disclosed
EP-2970265-B1 HETEROCYCLIC COMPOUNDS AND USES THEREOF PLEXXIKON INC (US) 2018-08-08 EP disclosed
US-20180072722-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF Opna Bio SA (CH) 2018-03-15 US disclosed
US-20180072722-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF Opna Bio SA (CH) 2018-03-15 US disclosed
US-20180072722-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF Opna Bio SA (CH) 2018-03-15 US disclosed
US-9822109-B2 Heterocyclic compounds and uses thereof PLEXXIKON INC. (US) 2017-11-21 US disclosed
US-9822109-B2 Heterocyclic compounds and uses thereof PLEXXIKON INC. (US) 2017-11-21 US disclosed
US-9822109-B2 Heterocyclic compounds and uses thereof PLEXXIKON INC. (US) 2017-11-21 US disclosed
US-20170320899-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF PLEXXIKON INC. (US) 2017-11-09 US disclosed
US-20160068528-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF Opna Bio SA (CH) 2016-03-10 US disclosed
US-20160068528-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF Opna Bio SA (CH) 2016-03-10 US disclosed
EP-2970265-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF PLEXXIKON INC. (US) 2016-01-20 EP disclosed
US-20150133400-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF Opna Bio SA (CH) 2015-05-14 US disclosed
US-20150133400-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF Opna Bio SA (CH) 2015-05-14 US disclosed
US-20150133400-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF Opna Bio SA (CH) 2015-05-14 US disclosed
US-20140303121-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF PLEXXIKON INC. 2014-10-09 US disclosed
US-20140303121-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF PLEXXIKON INC. 2014-10-09 US disclosed
US-20140303121-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF PLEXXIKON INC. 2014-10-09 US disclosed
WO-2014145051-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF ZHANG JIAZHONG (US) 2014-09-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140303121-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF CYP11B2, CYP11B1, CYP2C19 BRD4 1365/4885MEN1 672/4885KMT2A 4032/4885
US-20150133400-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF CYP11B2, CYP11B1, CYP2C19 BRD4 1365/4885MEN1 672/4885KMT2A 4032/4885
US-20170320899-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF CYP11B2, CYP11B1, CYP2C19 BRD4 1365/4885MEN1 672/4885KMT2A 4032/4885
US-20160068528-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF CYP11B2, CYP11B1, CYP2C19 BRD4 1365/4885MEN1 672/4885KMT2A 4032/4885
US-20180072722-A1 HETEROCYCLIC COMPOUNDS AND USES THEREOF CYP11B2, CYP11B1, CYP2C19 BRD4 1365/4885MEN1 672/4885KMT2A 4032/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.