SCHEMBL16065255

SCHEMBL16065255

CCCCCCOc1cc(-c2nc(C(=O)OC)co2)cc[n+]1O

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.38
HDAC8 Q9BY41 5/20 0.38
HDAC6 Q9UBN7 5/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
DAGLA Q9Y4D2 1/20 0.36
SMPD1 P17405 1/20 0.35
IRAK4 Q9NWZ3 2/20 0.35
ROCK2 O75116 1/20 0.34
ALPL P05186 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17412629 0.92 HDAC1 (0.38) HDAC1HDAC8HDAC6DAGLAIRAK4
SCHEMBL18723256 0.82 HDAC1 (0.37) HDAC1HDAC8HDAC6DAGLAIRAK4
SCHEMBL16065256 0.81 SMPD1 (0.41) HDAC1HDAC8HDAC6MAOAMAOB
SCHEMBL16065263 0.80 HDAC1 (0.36) HDAC1HDAC8HDAC6
SCHEMBL16065231 0.78 HDAC1 (0.44) HDAC1HDAC8HDAC6IRAK4ROCK2
SCHEMBL16748703 0.73 DAGLA (0.34) HDAC1HDAC8HDAC6MAOAMAOB
SCHEMBL17406937 0.72 IRAK4 (0.40) HDAC1HDAC8HDAC6DAGLAIRAK4
SCHEMBL18723160 0.72 IRAK4 (0.41) SMPD1IRAK4
SCHEMBL17407015 0.72 IRAK4 (0.41) SMPD1IRAK4
SCHEMBL12800496 0.71 HDAC1 (0.49) HDAC1HDAC8HDAC6DAGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014143672-A1 MACROCYCLIC COMPOUNDS AS IRAK4 INHIBITORS FOR THE TREATMENT OF INFLAMMATORY DISEASES BIOGEN IDEC MA INC. (US) 2014-09-18 WO disclosed