SCHEMBL16748703

SCHEMBL16748703

CCCCOc1cc(-c2nc(C(=O)OC)co2)[n+](O)cc1OCCCC

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAGLA Q9Y4D2 1/20 0.34
HDAC1 Q13547 2/20 0.33
HDAC8 Q9BY41 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
ALPL P05186 1/20 0.33
PLA2G2A P14555 2/20 0.33
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
TP53 P04637 4/20 0.32
SMPD1 P17405 3/20 0.32
TSHR P16473 3/20 0.32
GAA P10253 2/20 0.32
HTT P42858 1/20 0.32
CASP1 P29466 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16748705 0.90 TP53 (0.37) PDE4BPDE4DTP53NPC1RAB9A
SCHEMBL9915354 0.89 TP53 (0.33) DAGLAHDAC1HDAC8HDAC6MAOA
SCHEMBL9915361 0.80 ALPL (0.37) DAGLAHDAC1HDAC8HDAC6MAOA
SCHEMBL9915358 0.78 S1PR3 (0.37) TP53NPC1RAB9AKDM4EALDH1A1
SCHEMBL16748640 0.74 SMPD1 (0.38) ALPLPLA2G2APDE4APDE4BPDE4C
SCHEMBL16065255 0.73 HDAC1 (0.38) DAGLAHDAC1HDAC8HDAC6MAOA
SCHEMBL14124836 0.72 DAGLA (0.41) DAGLAHDAC1HDAC8HDAC6SMPD1
SCHEMBL16748687 0.71 HPGD (0.43) SMPD1HTTNPC1RAB9AALDH1A1
SCHEMBL16748690 0.71 MAPT (0.41) TP53SMPD1TSHRNPC1RAB9A
SCHEMBL16747529 0.70 XDH (0.41) TP53TSHRALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2646436-B1 MONOBACTAMS PFIZER (US) 2015-05-27 EP disclosed