Mifepristone

Mifepristone

SCHEMBL16087

CC#C[C@]1(O)CC[C@H]2[C@@H]3CCC4=CC(=O)CCC4=C3[C@@H](c3ccc(N(C)C)cc3)C[C@@]21C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

NR3C1PGR

The experimentally established mechanism targets of Mifepristone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 known ✓ P04150 10/20 1.00
PGR known ✓ P06401 10/20 1.00
AR P10275 5/20 1.00
CYP3A4 P08684 4/20 1.00
CYP2D6 P10635 3/20 1.00
CYP2C19 P33261 3/20 1.00
CYP2C9 P11712 3/20 1.00
CYP1A2 P05177 2/20 1.00
MAPK1 P28482 2/20 1.00
TDP1 Q9NUW8 2/20 1.00
LMNA P02545 2/20 1.00
MEN1 O00255 1/20 1.00
TP53 P04637 1/20 1.00
ALOX15 P16050 1/20 1.00
NFKB1 P19838 1/20 1.00
THPO P40225 1/20 1.00
KMT2A Q03164 1/20 1.00
NR1I2 O75469 1/20 1.00
GMNN O75496 1/20 1.00
ABCB11 O95342 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Mifepristone SCHEMBL19236544 1.00 NR3C1 (1.00) NR3C1PGRARCYP3A4CYP2D6
Mifepristone SCHEMBL13110930 1.00 NR3C1 (1.00) NR3C1PGRARCYP3A4CYP2D6
Mifepristone SCHEMBL19100510 1.00 NR3C1 (1.00) NR3C1PGRARCYP3A4CYP2D6
Mifepristone SCHEMBL13840946 1.00 NR3C1 (1.00) NR3C1PGRARCYP3A4CYP2D6
Mifepristone SCHEMBL10622661 1.00 NR3C1 (1.00) NR3C1PGRARCYP3A4CYP2D6
Mifepristone SCHEMBL10625406 1.00 NR3C1 (1.00) NR3C1PGRARCYP3A4CYP2D6
Mifepristone SCHEMBL10607607 1.00 NR3C1 (1.00) NR3C1PGRARCYP3A4CYP2D6
Mifepristone SCHEMBL918725 1.00 NR3C1 (1.00) NR3C1PGRARCYP3A4CYP2D6
Mifepristone SCHEMBL20769786 1.00 NR3C1 (1.00) NR3C1PGRARCYP3A4CYP2D6
Mifepristone SCHEMBL14870641 1.00 NR3C1 (1.00) NR3C1PGRARCYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 32868 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4747611-A1 OPTICAL ELECTRODE ANALYTE DETECTION SYSTEM AND METHODS OF USE Vital Biosciences Inc. (CA) 2026-05-27 EP claimed
CN-122094963-A Cardioprotective lipids and methods of use 2026-05-26 CN claimed
US-12629363-B2 Prophylaxis and treatment of angioedema PHARVARIS GMBH (CH) 2026-05-19 US claimed
US-20260130899-A1 METHOD OF TREATMENT FOR PREVENTION OF GLUCOCORTICOID TOXICITY AND/OR ENHANCEMENT OF MUSCLE REGENERATION VIA NEUTROPHIL ELASTASE INHIBITION THE RESEARCH FOUNDATION FOR THE STATE UNIVERSITY OF NEW YORK (US) 2026-05-14 US claimed
US-12625150-B2 Treatment of, and differential diagnosis between, ACTH-dependent Cushing's syndrome and ACTH-independent Cushing's syndrome CORCEPT THERAPEUTICS INCORPORATED (US) 2026-05-12 US claimed
US-12617809-B2 Cardioprotective lipid and method of use SIGNPATH PHARMA, INC. (US) 2026-05-05 US claimed
US-12616781-B2 Tubular nonwoven structure as active agent carrier for the atraumatic treatment of hollow organs, and a process for producing the same BVS—Best Vascular Solutions GmbH (DE) 2026-05-05 US claimed
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
US-20260115203-A1 LOW-DOSE MIFEPRISTONE FOR THE TREATMENT OF ENDOMETRIOSIS ASSOCIATED PAIN LABORATORIOS LITAPHAR S L (ES) 2026-04-30 US claimed
US-20260115317-A1 GENE THERAPY IMPERIAL COLLEGE INNOVATIONS LTD (GB) 2026-04-30 US claimed
EP-0266303-B1 ANTIGESTAGENS FOR THE INHIBITION OF UTERINE PROSTAGLANDIN SYNTHESIS SCHERING AKTIENGESELLSCHAFT (DE) 1992-07-29 EP claimed
EP-0446124-A2 Use of antiprogestomimetics to synchronise parturition in livestock ROUSSEL UCLAF (FR) 1991-09-11 EP claimed
EP-0184471-B1 PRODUCT CONTAINING AN ANTIPROGESTOMIMETIC AND A UTEROTONIC SUBSTANCE ROUSSEL-UCLAF (FR) 1990-11-14 EP claimed
US-4891368-A ESTRANE AND GONANE STEROIDS SCHERING AKTIENGESELLSCHAFT (DE) 1990-01-02 US claimed
US-4888331-A SIDE EFFECT REDUCTION; SCHERING AKTIENGESELLSCHAFT (DE) 1989-12-19 US claimed
EP-0135400-B1 ESTRADIENE DERIVATIVES LABELLED WITH TRITIUM, THEIR PREPARATION AND INTERMEDIATES FOR THEIR PREPARATION, AND THEIR UTILIZATION IN THE STUDY AND IN THE DETERMINATION OF STEROIDS IN BIOLOGICAL FLUIDS ROUSSEL-UCLAF (FR) 1988-06-01 EP claimed
EP-0139608-B1 PROSTAGLANDINS AND ANTIGESTAGENS FOR THE ONSET OF LABOUR OR FOR THE INTERRUPTION OF PREGNANCY SCHERING AKTIENGESELLSCHAFT (DE) 1988-06-01 EP claimed
EP-0135400-A2 Estradiene derivatives labelled with tritium, their preparation and intermediates for their preparation, and their utilization in the study and in the determination of steroids in biological fluids ROUSSEL-UCLAF (FR) 1985-03-27 EP claimed
EP-0057115-B1 STEROID DERIVATIVES SUBSTITUTED IN THE 11-BETA POSITION, PROCESS FOR THEIR PREPARATION, THEIR UTILIZATION AS MEDICAMENTS AND COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1985-03-20 EP claimed
EP-0131491-A1 Estradiene derivatives labelled with iodine, process for their preparation and intermediates in their preparation, and their use in the study and the radioimmunological determination of steroids in body fluids ROUSSEL-UCLAF (FR) 1985-01-16 EP claimed