SCHEMBL16087516

SCHEMBL16087516

CCc1cc([C@H]2CC[C@@H](c3nnc4n3-c3ccc(Cl)cc3CN(OC(=O)OC(C)(C)C)C4)CC2)no1

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 19/20 0.50
KCNH2 Q12809 7/20 0.50
OXTR P30559 2/20 0.47
AVPR2 P30518 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16087505 1.00 AVPR1A (0.50) AVPR1AKCNH2OXTRAVPR2
SCHEMBL16087513 0.91 AVPR1A (0.62) AVPR1AKCNH2OXTRAVPR2
SCHEMBL2585593 0.88 OXTR (0.56) AVPR1AKCNH2OXTRAVPR2
SCHEMBL2588113 0.88 OXTR (0.56) AVPR1AKCNH2OXTRAVPR2
SCHEMBL2585590 0.88 OXTR (0.56) AVPR1AKCNH2OXTRAVPR2
SCHEMBL16087561 0.87 AVPR1A (0.47) AVPR1AKCNH2OXTRAVPR2
SCHEMBL16087519 0.87 AVPR1A (0.47) AVPR1AKCNH2OXTRAVPR2
SCHEMBL11890017 0.85 AVPR1A (0.51) AVPR1AKCNH2OXTRAVPR2
SCHEMBL16774898 0.85 AVPR1A (0.47) AVPR1AKCNH2OXTRAVPR2
SCHEMBL16087524 0.84 AVPR1A (0.49) AVPR1AKCNH2OXTRAVPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2569319-B1 HETEROARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES HOFFMANN LA ROCHE (CH) 2014-09-24 EP claimed