SCHEMBL16092209

SCHEMBL16092209

Nc1cc(-c2ccncc2)c(Cl)nn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
GFER P55789 1/20 0.44
CASP1 P29466 2/20 0.42
CCNC P24863 2/20 0.39
CDK8 P49336 2/20 0.39
AAK1 Q2M2I8 1/20 0.38
ATAD2 Q6PL18 1/20 0.38
LMNA P02545 2/20 0.37
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
AURKB Q96GD4 1/20 0.37
INCENP Q9NQS7 1/20 0.37
IMPDH2 P12268 1/20 0.37
GCGR P47871 1/20 0.37
MAPK14 Q16539 1/20 0.37
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL526496 0.82 SMARCA2 (0.46) SMN1; SMN2NPC1RAB9ACASP1LMNA
SCHEMBL2646929 0.80 CASP1 (0.41) MAPTSMN1; SMN2NPC1RAB9AGFER
SCHEMBL30453161 0.80 CASP1 (0.41) MAPTSMN1; SMN2NPC1RAB9AGFER
SCHEMBL1038525 0.79 CASP1 (0.48) NPC1RAB9ACASP1
SCHEMBL19440997 0.77 CASP1 (0.40) MAPTSMN1; SMN2NPC1RAB9AGFER
SCHEMBL19813305 0.77 CYP2A6 (0.44) MAPTIMPDH2ALDH1A1
SCHEMBL28685605 0.75 CASP1 (0.48) MAPTSMN1; SMN2NPC1RAB9ACASP1
SCHEMBL1754688 0.74 MAPK1 (0.53) MAPTNPC1RAB9ACASP1ATAD2
SCHEMBL16061219 0.73 MAPK14 (0.60) MAPTSMN1; SMN2NPC1RAB9AGFER
SCHEMBL16092109 0.73 CASP1 (0.43) MAPTSMN1; SMN2NPC1RAB9AGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014145485-A2 MAP KINASE MODULATORS AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2014-09-18 WO disclosed