SCHEMBL16093333

SCHEMBL16093333

NC(=O)[C@@H](N)Cc1ccc(S(N)(=O)=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA2 P00918 18/20 0.54
CA1 P00915 12/20 0.54
KDM4E B2RXH2 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
CA12 O43570 8/20 0.53
CA9 Q16790 7/20 0.53
CA4 P22748 5/20 0.53
CA6 P23280 5/20 0.53
CA5A P35218 5/20 0.53
CA7 P43166 5/20 0.53
CA14 Q9ULX7 5/20 0.53
CA5B Q9Y2D0 5/20 0.53
CA3 P07451 1/20 0.51
CA13 Q8N1Q1 1/20 0.51
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19941420 1.00 CA2 (0.54) CA2CA1KDM4ESMN1; SMN2CA12
SCHEMBL30998999 0.86 SLC7A5 (0.62) CA2CA1KDM4ESMN1; SMN2CA12
SCHEMBL18926112 0.84 EPHX1 (0.51) KDM4ESMN1; SMN2
SCHEMBL10251218 0.84 EPHX1 (0.51) KDM4ESMN1; SMN2
SCHEMBL2072326 0.83 SLC7A5 (0.53) CA2CA1CA12
SCHEMBL2072328 0.83 SLC7A5 (0.53) CA2CA1CA12
SCHEMBL27734534 0.81 SLC7A5 (0.57) CA2CA1KDM4ESMN1; SMN2CA12
SCHEMBL19938091 0.81 CA2 (0.53) CA2CA1KDM4ESMN1; SMN2CA12
SCHEMBL15881217 0.81 CA2 (0.53) CA2CA1KDM4ESMN1; SMN2CA12
SCHEMBL6951101 0.78 CA2 (0.62) CA2CA1KDM4ESMN1; SMN2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8841263-B2 Macrocyclic compounds and methods of making and using the same MELINTA THERAPEUTICS, INC. (US) 2014-09-23 US disclosed