SCHEMBL1609640

SCHEMBL1609640

COc1ccc(C(=O)CNC(=O)c2cc3cc(Cl)ccc3[nH]2)cc1

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 2/20 0.60
PYGL P06737 12/20 0.57
HRH4 Q9H3N8 1/20 0.56
HRH3 Q9Y5N1 1/20 0.56
KDM4E B2RXH2 2/20 0.55
MEN1 O00255 1/20 0.55
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
KMT2A Q03164 1/20 0.55
ALDH1A1 P00352 1/20 0.55
MAPT P10636 1/20 0.55
PDGFRB P09619 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2107375 0.84 KDM4E (0.47) PYGLKDM4EMEN1NPC1RAB9A
SCHEMBL6398667 0.84 MAPT (0.67) FLT3KDM4EMEN1NPC1RAB9A
SCHEMBL1608132 0.83 PYGL (0.57) PYGLHRH4HRH3
SCHEMBL6162398 0.82 PYGL (0.69) PYGLHRH4HRH3
SCHEMBL1608140 0.82 PYGL (0.59) PYGLHRH4HRH3MEN1KMT2A
SCHEMBL1608567 0.81 GUSB (0.60) PYGLHRH4HRH3
SCHEMBL3253089 0.78 PYGL (0.67) FLT3PYGLHRH4HRH3
SCHEMBL4919678 0.78 FLT3 (0.61) FLT3PYGLHRH4HRH3KDM4E
SCHEMBL5891883 0.78 PYGL (0.67) PYGLHRH4HRH3
SCHEMBL23014105 0.78 KMT2A (0.60) KDM4EMEN1NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110086885-A1 Indole-2-carboxylic acid amides PROSIDION LIMITED (GB) 2011-04-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110086885-A1 Indole-2-carboxylic acid amides IDO2, IDO1, CPT1A FLT3 2303/4885PYGL 152/4885HRH4 676/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.