SCHEMBL16098091

SCHEMBL16098091

O=C(O)C1CCC(=O)N1c1nc(Cl)ncc1F

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
ABL1 P00519 2/20 0.35
BCR P11274 2/20 0.35
KMT2A Q03164 1/20 0.35
RPS6KA5 O75582 1/20 0.34
P2RX7 Q99572 8/20 0.34
HDAC1 Q13547 3/20 0.32
HDAC8 Q9BY41 3/20 0.32
HDAC6 Q9UBN7 3/20 0.32
ACE P12821 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16097228 0.80 SMN1; SMN2 (0.41) MAPTSMN1; SMN2HCRTR1HCRTR2ABL1
SCHEMBL16097225 0.80 SMN1; SMN2 (0.41) MAPTSMN1; SMN2HCRTR1HCRTR2ABL1
SCHEMBL9104817 0.72 HDAC1 (0.42) MAPTSMN1; SMN2HCRTR1HDAC1HDAC8
SCHEMBL9104794 0.72 HDAC1 (0.42) MAPTSMN1; SMN2HCRTR1HDAC1HDAC8
SCHEMBL3710014 0.72 P2RX7 (0.39) P2RX7ACE
SCHEMBL3710013 0.72 P2RX7 (0.39) P2RX7ACE
SCHEMBL2568372 0.72 NPC1 (0.51) MAPTSMN1; SMN2KMT2A
SCHEMBL2568370 0.72 NPC1 (0.51) MAPTSMN1; SMN2KMT2A
SCHEMBL16098502 0.70 MAPT (0.41) MAPTSMN1; SMN2HCRTR1HCRTR2KMT2A
SCHEMBL16098503 0.70 MAPT (0.41) MAPTSMN1; SMN2HCRTR1HCRTR2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014147586-A1 1-(2-(ETHYLAMINO)PYRIMIDIN-4-YL)PYRROLIDIN-2-ONES AS INHIBITORS OF MUTANT IDH NOVARTIS AG (CH) 2014-09-25 WO disclosed