SCHEMBL16099754

SCHEMBL16099754

COc1cc(C)c2c3ccncc3n(CCN3CCOCC3)c2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HASPIN Q8TF76 1/20 0.45
NFATC1 O95644 1/20 0.41
GSK3B P49841 1/20 0.41
DYRK1A Q13627 1/20 0.41
CNR1 P21554 2/20 0.41
ALDH1A1 P00352 4/20 0.41
TSHR P16473 2/20 0.41
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CNR2 P34972 1/20 0.41
RECQL P46063 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
LMNA P02545 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
ATM Q13315 1/20 0.39
HSD17B10 Q99714 1/20 0.39
PDE5A O76074 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16099021 0.95 HASPIN (0.47) HASPINNFATC1GSK3BDYRK1AALDH1A1
SCHEMBL16099658 0.85 NFATC1 (0.43) NFATC1GSK3BDYRK1ATSHRLMNA
SCHEMBL16093883 0.82 PDE5A (0.37) NFATC1GSK3BDYRK1AALDH1A1LMNA
SCHEMBL16098852 0.81 HASPIN (0.45) HASPINNFATC1GSK3BDYRK1AALDH1A1
SCHEMBL16098887 0.80 HASPIN (0.66) HASPINDYRK1ATSHRTP53CYP1A2
SCHEMBL16099514 0.80 DYRK1A (0.49) HASPINDYRK1AALDH1A1TP53CYP1A2
SCHEMBL16093943 0.80 NFATC1 (0.47) NFATC1GSK3BDYRK1ACYP3A4KDM4E
SCHEMBL16093779 0.79 HASPIN (0.71) HASPINDYRK1ATP53CYP1A2CYP3A4
SCHEMBL16099752 0.78 HASPIN (0.47) HASPINDYRK1AALDH1A1TP53CYP1A2
SCHEMBL16098427 0.76 HASPIN (0.43) HASPINDYRK1ATP53CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2968284-A2 ALKYL-AMINE HARMINE DERIVATIVES FOR PROMOTING BONE GROWTH Osteoqc Inc. (CA) 2016-01-20 EP disclosed
WO-2014153203-A2 ALKYL-AMINE HARMINE DERIVATIVES FOR PROMOTING BONE GROWTH OSSIFI INC. (US) 2014-09-25 WO disclosed