SCHEMBL16104652

SCHEMBL16104652

CC(C)(C)CCC(=O)N1CCC(N)(C#N)CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.35
NPC1 O15118 2/20 0.34
KDM1A O60341 1/20 0.32
ITGB3 P05106 2/20 0.31
ITGA2B P08514 2/20 0.31
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31
APH1B Q8WW43 1/20 0.31
NCSTN Q92542 1/20 0.31
APH1A Q96BI3 1/20 0.31
PSENEN Q9NZ42 1/20 0.31
ATM Q13315 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
USP2 O75604 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
CYP3A4 P08684 1/20 0.31
HPGD P15428 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26802659 0.74 ALDH1A1 (0.34) NPC1ITGB3ITGA2BATMKDM4E
SCHEMBL6836951 0.73 CYP2C9 (0.40) KDM4EMEN1USP2ALDH1A1CYP3A4
SCHEMBL5356389 0.73 CYP2C9 (0.40) KDM4EMEN1USP2ALDH1A1CYP3A4
SCHEMBL19169730 0.73 ATM (0.52) NPC1ATMKDM4EMEN1USP2
SCHEMBL13839275 0.73 ATM (0.58) NPC1ATMKDM4EMEN1USP2
SCHEMBL6356887 0.72 DPP4 (0.34) DPP4
SCHEMBL849908 0.72 USP2 (0.47) MEN1USP2ALDH1A1HPGDKMT2A
SCHEMBL2739384 0.71 ATM (0.56) NPC1ATMMEN1ALDH1A1CYP3A4
SCHEMBL850964 0.71 CA12 (0.35)
SCHEMBL1140258 0.70 ALDH1A1 (0.49) ATMKDM4EMEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2433940-B1 SPIROIMIDAZOLONE DERIVATIVE CHUGAI PHARMACEUTICAL CO LTD (JP) 2014-09-24 EP disclosed
EP-2433940-A1 SPIROIMIDAZOLONE DERIVATIVE Chugai Seiyaku Kabushiki Kaisha (JP) 2012-03-28 EP disclosed